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Kelly Chibale

Showing results (131-140 of 315) with videos related to

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Bioorganic & Medicinal Chemistry Letters|July 4, 2012
Benzoheterocyclic amodiaquine analogues with potent antiplasmodial activity: synthesis and pharmacological evaluationDennis S B Ongarora, Jiri Gut, Philip J Rosenthal, et al.
Malaria Journal|February 7, 2014
CRIMALDDI: platform technologies and novel anti-malarial drug targetsHenri Vial, Donatella Taramelli, Ian C Boulton, et al.
Bioorganic & Medicinal Chemistry Letters|October 24, 2007
Design, synthesis, and antimalarial activity of structural chimeras of thiosemicarbazone and ferroquine analoguesChristophe Biot, Bruno Pradines, Marie-Hélène Sergeant, et al.
European Journal of Medicinal Chemistry|June 27, 2015
Synthesis, antiplasmodial activity and mechanistic studies of pyrimidine-5-carbonitrile and quinoline hybridsHardeep Kaur, Jan Balzarini, Carmen de Kock, et al.
Nature Communications|September 15, 2023
First fully-automated AI/ML virtual screening cascade implemented at a drug discovery centre in AfricaGemma Turon, Jason Hlozek, John G Woodland, et al.
Bioorganic & Medicinal Chemistry Letters|April 22, 2011
Synthesis and in vitro antitubercular activity of ferrocene-based hydrazonesAman Mahajan, Laurent Kremer, Stefan Louw, et al.
International Journal of Antimicrobial Agents|July 13, 2005
Reversal of chloroquine resistance in Plasmodium falciparum by 9H-xanthene derivativesChung-Pu Wu, Donelly A van Schalkwyk, Dale Taylor, et al.
Drug Metabolism and Personalized Therapy|October 9, 2016
Improvement of the chemical inhibition phenotyping assay by cross-reactivity correctionNicholas M Njuguna, Ken-Ichi Umehara, Felix Huth, et al.
Journal of Pharmaceutical Sciences|March 1, 2019
Cocrystal and Salt Forms of an Imidazopyridazine Antimalarial Drug LeadTerence J Noonan, Kelly Chibale, Peter M Cheuka, et al.
European Journal of Medicinal Chemistry|July 6, 2015
Primaquine-pyrimidine hybrids: synthesis and dual-stage antiplasmodial activityHardeep Kaur, Marta Machado, Carmen de Kock, et al.
Pageof 32

Showing results (131-140 of 315) with videos related to

Sort By:
Pageof 32
Bioorganic & Medicinal Chemistry Letters|July 4, 2012
Benzoheterocyclic amodiaquine analogues with potent antiplasmodial activity: synthesis and pharmacological evaluationDennis S B Ongarora, Jiri Gut, Philip J Rosenthal, et al.
Malaria Journal|February 7, 2014
CRIMALDDI: platform technologies and novel anti-malarial drug targetsHenri Vial, Donatella Taramelli, Ian C Boulton, et al.
Bioorganic & Medicinal Chemistry Letters|October 24, 2007
Design, synthesis, and antimalarial activity of structural chimeras of thiosemicarbazone and ferroquine analoguesChristophe Biot, Bruno Pradines, Marie-Hélène Sergeant, et al.
European Journal of Medicinal Chemistry|June 27, 2015
Synthesis, antiplasmodial activity and mechanistic studies of pyrimidine-5-carbonitrile and quinoline hybridsHardeep Kaur, Jan Balzarini, Carmen de Kock, et al.
Nature Communications|September 15, 2023
First fully-automated AI/ML virtual screening cascade implemented at a drug discovery centre in AfricaGemma Turon, Jason Hlozek, John G Woodland, et al.
Bioorganic & Medicinal Chemistry Letters|April 22, 2011
Synthesis and in vitro antitubercular activity of ferrocene-based hydrazonesAman Mahajan, Laurent Kremer, Stefan Louw, et al.
International Journal of Antimicrobial Agents|July 13, 2005
Reversal of chloroquine resistance in Plasmodium falciparum by 9H-xanthene derivativesChung-Pu Wu, Donelly A van Schalkwyk, Dale Taylor, et al.
Drug Metabolism and Personalized Therapy|October 9, 2016
Improvement of the chemical inhibition phenotyping assay by cross-reactivity correctionNicholas M Njuguna, Ken-Ichi Umehara, Felix Huth, et al.
Journal of Pharmaceutical Sciences|March 1, 2019
Cocrystal and Salt Forms of an Imidazopyridazine Antimalarial Drug LeadTerence J Noonan, Kelly Chibale, Peter M Cheuka, et al.
European Journal of Medicinal Chemistry|July 6, 2015
Primaquine-pyrimidine hybrids: synthesis and dual-stage antiplasmodial activityHardeep Kaur, Marta Machado, Carmen de Kock, et al.
Pageof 32