Jove
Visualize
Contact Us
JoVE
x logofacebook logolinkedin logoyoutube logo
ABOUT JoVE
OverviewLeadershipBlogJoVE Help Center
AUTHORS
Publishing ProcessEditorial BoardScope & PoliciesPeer ReviewFAQSubmit
LIBRARIANS
TestimonialsSubscriptionsAccessResourcesLibrary Advisory BoardFAQ
RESEARCH
JoVE JournalMethods CollectionsJoVE Encyclopedia of ExperimentsArchive
EDUCATION
JoVE CoreJoVE BusinessJoVE Science EducationJoVE Lab ManualFaculty Resource CenterFaculty Site
Terms & Conditions of Use
Privacy Policy
Policies

Filters

Kelly Chibale

Showing results (301-310 of 315) with videos related to

Pageof 32
Sort By:
Science Translational Medicine|October 19, 2022
The anticancer human mTOR inhibitor sapanisertib potently inhibits multiple <i>Plasmodium</i> kinases and life cycle stagesLauren B Arendse, James M Murithi, Tarrick Qahash, et al.
Cell Chemical Biology|May 4, 2020
Inhibition of Resistance-Refractory P. falciparum Kinase PKG Delivers Prophylactic, Blood Stage, and Transmission-Blocking Antiplasmodial ActivityManu Vanaerschot, James M Murithi, Charisse Flerida A Pasaje, et al.
Nature Communications|January 12, 2021
Multistage and transmission-blocking targeted antimalarials discovered from the open-source MMV Pandemic Response BoxJanette Reader, Mariëtte E van der Watt, Dale Taylor, et al.
ACS Infectious Diseases|March 10, 2018
2-Mercapto-Quinazolinones as Inhibitors of Type II NADH Dehydrogenase and Mycobacterium tuberculosis: Structure-Activity Relationships, Mechanism of Action and Absorption, Distribution, Metabolism, and Excretion CharacterizationDinakaran Murugesan, Peter C Ray, Tracy Bayliss, et al.
Biorxiv : the Preprint Server for Biology|August 12, 2025
The Human Chk1 Inhibitor CHIR-124 Shows Multistage Activity Against <i>Plasmodium falciparum</i> via Dual Inhibition of <i>Pf</i>Ark1 and Hemozoin FormationKathryn J Wicht, John G Woodland, Larnelle F Garnie, et al.
Angewandte Chemie (International Ed. in English)|May 3, 2025
The ATM Kinase Inhibitor AZD0156 Is a Potent Inhibitor of Plasmodium Phosphatidylinositol 4-Kinase (PI4Kβ) and Is an Attractive Candidate for Medicinal Chemistry Optimization Against MalariaJohn G Woodland, Dina Coertzen, Kathryn J Wicht, et al.
ACS Chemical Biology|June 13, 2026
The Human Chk1 Inhibitor CHIR-124 Shows Multistage Activity against the Human Malaria Parasite <i>Plasmodium falciparum</i> via Polypharmacological Inhibition of <i>Pf</i>Ark1 and Hemozoin FormationKathryn J Wicht, John G Woodland, Larnelle F Garnie, et al.
Cell Chemical Biology|July 7, 2021
The Plasmodium falciparum ABC transporter ABCI3 confers parasite strain-dependent pleiotropic antimalarial drug resistanceJames M Murithi, Ioanna Deni, Charisse Flerida A Pasaje, et al.
Journal of Medicinal Chemistry|November 18, 2017
Novel Antitubercular 6-Dialkylaminopyrimidine Carboxamides from Phenotypic Whole-Cell High Throughput Screening of a SoftFocus Library: Structure-Activity Relationship and Target Identification StudiesColin R Wilson, Richard K Gessner, Atica Moosa, et al.
Journal of Medicinal Chemistry|June 25, 2024
2,8-Disubstituted-1,5-naphthyridines as Dual Inhibitors of <i>Plasmodium falciparum</i> Phosphatidylinositol-4-kinase and Hemozoin Formation with <i>In Vivo</i> EfficacyGodwin Akpeko Dziwornu, Donald Seanego, Stephen Fienberg, et al.
Pageof 32

Showing results (301-310 of 315) with videos related to

Sort By:
Pageof 32
Science Translational Medicine|October 19, 2022
The anticancer human mTOR inhibitor sapanisertib potently inhibits multiple <i>Plasmodium</i> kinases and life cycle stagesLauren B Arendse, James M Murithi, Tarrick Qahash, et al.
Cell Chemical Biology|May 4, 2020
Inhibition of Resistance-Refractory P. falciparum Kinase PKG Delivers Prophylactic, Blood Stage, and Transmission-Blocking Antiplasmodial ActivityManu Vanaerschot, James M Murithi, Charisse Flerida A Pasaje, et al.
Nature Communications|January 12, 2021
Multistage and transmission-blocking targeted antimalarials discovered from the open-source MMV Pandemic Response BoxJanette Reader, Mariëtte E van der Watt, Dale Taylor, et al.
ACS Infectious Diseases|March 10, 2018
2-Mercapto-Quinazolinones as Inhibitors of Type II NADH Dehydrogenase and Mycobacterium tuberculosis: Structure-Activity Relationships, Mechanism of Action and Absorption, Distribution, Metabolism, and Excretion CharacterizationDinakaran Murugesan, Peter C Ray, Tracy Bayliss, et al.
Biorxiv : the Preprint Server for Biology|August 12, 2025
The Human Chk1 Inhibitor CHIR-124 Shows Multistage Activity Against <i>Plasmodium falciparum</i> via Dual Inhibition of <i>Pf</i>Ark1 and Hemozoin FormationKathryn J Wicht, John G Woodland, Larnelle F Garnie, et al.
Angewandte Chemie (International Ed. in English)|May 3, 2025
The ATM Kinase Inhibitor AZD0156 Is a Potent Inhibitor of Plasmodium Phosphatidylinositol 4-Kinase (PI4Kβ) and Is an Attractive Candidate for Medicinal Chemistry Optimization Against MalariaJohn G Woodland, Dina Coertzen, Kathryn J Wicht, et al.
ACS Chemical Biology|June 13, 2026
The Human Chk1 Inhibitor CHIR-124 Shows Multistage Activity against the Human Malaria Parasite <i>Plasmodium falciparum</i> via Polypharmacological Inhibition of <i>Pf</i>Ark1 and Hemozoin FormationKathryn J Wicht, John G Woodland, Larnelle F Garnie, et al.
Cell Chemical Biology|July 7, 2021
The Plasmodium falciparum ABC transporter ABCI3 confers parasite strain-dependent pleiotropic antimalarial drug resistanceJames M Murithi, Ioanna Deni, Charisse Flerida A Pasaje, et al.
Journal of Medicinal Chemistry|November 18, 2017
Novel Antitubercular 6-Dialkylaminopyrimidine Carboxamides from Phenotypic Whole-Cell High Throughput Screening of a SoftFocus Library: Structure-Activity Relationship and Target Identification StudiesColin R Wilson, Richard K Gessner, Atica Moosa, et al.
Journal of Medicinal Chemistry|June 25, 2024
2,8-Disubstituted-1,5-naphthyridines as Dual Inhibitors of <i>Plasmodium falciparum</i> Phosphatidylinositol-4-kinase and Hemozoin Formation with <i>In Vivo</i> EfficacyGodwin Akpeko Dziwornu, Donald Seanego, Stephen Fienberg, et al.
Pageof 32