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Molecular Diversity
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November 7, 2019
Structure elaboration of isoniazid: synthesis, in silico molecular docking and antimycobacterial activity of isoniazid-pyrimidine conjugates
Hardeep Kaur, Lovepreet Singh, Kelly Chibale, et al.
Medchemcomm
|
August 16, 2018
Identification of steroid-like natural products as antiplasmodial agents by 2D and 3D similarity-based virtual screening
Elumalai Pavadai, Gurminder Kaur, Sergio Wittlin, et al.
ACS Infectious Diseases
|
December 25, 2018
Structure-Activity Relationship and in Vitro Absorption, Distribution, Metabolism, Excretion, and Toxicity (ADMET) Studies of N-aryl 3-Trifluoromethyl Pyrido[1,2- a]benzimidazoles That Are Efficacious in a Mouse Model of Schistosomiasis
Godfrey Mayoka, Jennifer Keiser, Cécile Häberli, et al.
Expert Opinion on Drug Metabolism & Toxicology
|
September 16, 2014
Physicochemical and drug metabolism characterization of a series of 4-aminoquinoline-3-hydroxypyridin-4-one hybrid molecules with antimalarial activity
Roslyn Thelingwani, Britta Bonn, Kelly Chibale, et al.
Journal of Chemical Information and Modeling
|
July 25, 2018
3D-QSAR Modeling and Synthesis of New Fusidic Acid Derivatives as Antiplasmodial Agents
Gurminder Kaur, Elumalai Pavadai, Sergio Wittlin, et al.
Molecules (Basel, Switzerland)
|
December 18, 2020
Synthesis and In Vitro Antiprotozoan Evaluation of 4-/8-Aminoquinoline-based Lactams and Tetrazoles
Matshawandile Tukulula, Stefan Louw, Mathew Njoroge, et al.
Journal of Pharmaceutical Sciences
|
September 20, 2016
Preparation and Physicochemical Characterization of an Inclusion Complex Between Dimethylated β-Cyclodextrin and a Drug Lead From a New Class of Orally Active Antimalarial 3,5-Diaryl-2-Aminopyridines
Laurelle M Joseph, Kelly Chibale, Mino R Caira
Bioorganic & Medicinal Chemistry Letters
|
May 24, 2005
Exploiting a basic chemosensitizing pharmacophore hypothesis. Part 1: synthesis and biological evaluation of novel arylbromide and bicyclic chemosensitizers against drug-resistant malaria parasites
Franck Chouteau, David Ramanitrahasimbola, Philippe Rasoanaivo, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 26, 2009
Synthesis and evaluation of phenylequine for antimalarial activity in vitro and in vivo
Margaret A L Blackie, Vanessa Yardley, Kelly Chibale
Bioorganic & Medicinal Chemistry Letters
|
June 30, 2014
Kojic acid derived hydroxypyridinone-chloroquine hybrids: synthesis, crystal structure, antiplasmodial activity and β-haematin inhibition
Warren Andrew Andayi, Timothy J Egan, Kelly Chibale
Page
of 32
Search research articles
Search
Showing results (41-50 of 315) with videos related to
Sort By:
Page
of 32
Molecular Diversity
|
November 7, 2019
Structure elaboration of isoniazid: synthesis, in silico molecular docking and antimycobacterial activity of isoniazid-pyrimidine conjugates
Hardeep Kaur, Lovepreet Singh, Kelly Chibale, et al.
Medchemcomm
|
August 16, 2018
Identification of steroid-like natural products as antiplasmodial agents by 2D and 3D similarity-based virtual screening
Elumalai Pavadai, Gurminder Kaur, Sergio Wittlin, et al.
ACS Infectious Diseases
|
December 25, 2018
Structure-Activity Relationship and in Vitro Absorption, Distribution, Metabolism, Excretion, and Toxicity (ADMET) Studies of N-aryl 3-Trifluoromethyl Pyrido[1,2- a]benzimidazoles That Are Efficacious in a Mouse Model of Schistosomiasis
Godfrey Mayoka, Jennifer Keiser, Cécile Häberli, et al.
Expert Opinion on Drug Metabolism & Toxicology
|
September 16, 2014
Physicochemical and drug metabolism characterization of a series of 4-aminoquinoline-3-hydroxypyridin-4-one hybrid molecules with antimalarial activity
Roslyn Thelingwani, Britta Bonn, Kelly Chibale, et al.
Journal of Chemical Information and Modeling
|
July 25, 2018
3D-QSAR Modeling and Synthesis of New Fusidic Acid Derivatives as Antiplasmodial Agents
Gurminder Kaur, Elumalai Pavadai, Sergio Wittlin, et al.
Molecules (Basel, Switzerland)
|
December 18, 2020
Synthesis and In Vitro Antiprotozoan Evaluation of 4-/8-Aminoquinoline-based Lactams and Tetrazoles
Matshawandile Tukulula, Stefan Louw, Mathew Njoroge, et al.
Journal of Pharmaceutical Sciences
|
September 20, 2016
Preparation and Physicochemical Characterization of an Inclusion Complex Between Dimethylated β-Cyclodextrin and a Drug Lead From a New Class of Orally Active Antimalarial 3,5-Diaryl-2-Aminopyridines
Laurelle M Joseph, Kelly Chibale, Mino R Caira
Bioorganic & Medicinal Chemistry Letters
|
May 24, 2005
Exploiting a basic chemosensitizing pharmacophore hypothesis. Part 1: synthesis and biological evaluation of novel arylbromide and bicyclic chemosensitizers against drug-resistant malaria parasites
Franck Chouteau, David Ramanitrahasimbola, Philippe Rasoanaivo, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 26, 2009
Synthesis and evaluation of phenylequine for antimalarial activity in vitro and in vivo
Margaret A L Blackie, Vanessa Yardley, Kelly Chibale
Bioorganic & Medicinal Chemistry Letters
|
June 30, 2014
Kojic acid derived hydroxypyridinone-chloroquine hybrids: synthesis, crystal structure, antiplasmodial activity and β-haematin inhibition
Warren Andrew Andayi, Timothy J Egan, Kelly Chibale
Page
of 32