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Plos One|July 26, 2017
Bruton's tyrosine kinase inhibitor BMS-986142 in experimental models of rheumatoid arthritis enhances efficacy of agents representing clinical standard-of-careKathleen M Gillooly, Claudine Pulicicchio, Mark A Pattoli, et al.Bioorganic & Medicinal Chemistry Letters|March 25, 2008
Pyrazolo-pyrimidines: a novel heterocyclic scaffold for potent and selective p38 alpha inhibitorsJagabandhu Das, Robert V Moquin, Sidney Pitt, et al.Bioorganic & Medicinal Chemistry Letters|June 2, 2007
Synthesis and structure-activity relationship of imidazo(1,2-a)thieno(3,2-e)pyrazines as IKK-beta inhibitorsMakonen Belema, Amy Bunker, Van N Nguyen, et al.The Journal of Pharmacology and Experimental Therapeutics|April 15, 2006
Selective inhibition of eosinophil influx into the lung by small molecule CC chemokine receptor 3 antagonists in mouse models of allergic inflammationAnuk M Das, Krishna G Vaddi, Kimberly A Solomon, et al.Journal of Leukocyte Biology|August 5, 2006
A selective small molecule agonist of the melanocortin-1 receptor inhibits lipopolysaccharide-induced cytokine accumulation and leukocyte infiltration in miceLiya Kang, Kim W McIntyre, Kathleen M Gillooly, et al.Journal of Medicinal Chemistry|May 16, 2003
Rational design and synthesis of an orally active indolopyridone as a novel conformationally constrained cannabinoid ligand possessing antiinflammatory propertiesStephen T Wrobleski, Ping Chen, John Hynes, et al.Bioorganic & Medicinal Chemistry Letters|February 17, 2006
Discovery and SAR of 2-amino-5-[(thiomethyl)aryl]thiazoles as potent and selective Itk inhibitorsJagabandhu Das, Chunjian Liu, Robert V Moquin, et al.Bioorganic & Medicinal Chemistry Letters|April 21, 2009
Synthesis, initial SAR and biological evaluation of 1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-4-amine derived inhibitors of IkappaB kinaseJames Kempson, Junqing Guo, Jagabandhu Das, et al.Bioorganic & Medicinal Chemistry Letters|November 18, 2004
Discovery of novel 2-(aminoheteroaryl)-thiazole-5-carboxamides as potent and orally active Src-family kinase p56(Lck) inhibitorsPing Chen, Derek Norris, Jagabandhu Das, et al.Bioorganic & Medicinal Chemistry Letters|November 2, 2010
5-amino-pyrazoles as potent and selective p38α inhibitorsJagabandhu Das, Robert V Moquin, Alaric J Dyckman, et al.Pageof 7