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Yakugaku Zasshi : Journal of the Pharmaceutical Society of Japan
|
October 1, 2025
[Development of Mid-size Bivalent Inhibitors Targeting a Cancer-related Kinase]
Kohei Tsuji
Bioorganic & Medicinal Chemistry
|
July 3, 2024
Design, synthesis and evaluation of bioactivity of peptidomimetics based on chloroalkene dipeptide isosteres
Takuya Kobayakawa, Kohei Tsuji, Hirokazu Tamamura
Bioorganic & Medicinal Chemistry
|
January 7, 2025
Fine-tuning probes for fluorescence polarization binding assays of bivalent ligands against polo-like kinase 1 using full-length protein
Kohei Tsuji, Hirokazu Tamamura, Terrence R Burke
Biological & Pharmaceutical Bulletin
|
July 10, 2024
Application of a Fluorescence Recovery-Based Polo-Like Kinase 1 Binding Assay to Polo-Like Kinase 2 and Polo-Like Kinase 3
Kohei Tsuji, Hirokazu Tamamura, Terrence R Burke
RSC Chemical Biology
|
August 2, 2024
Affinity enhancement of polo-like kinase 1 polo box domain-binding ligands by a bivalent approach using a covalent kinase-binding component
Kohei Tsuji, Hirokazu Tamamura, Terrence R Burke
Analytical Methods : Advancing Methods and Applications
|
September 24, 2020
A new genre of fluorescence recovery assay to evaluate polo-like kinase 1 ATP-competitive inhibitors
Kohei Tsuji, David Hymel, Terrence R Burke
Chemsuschem
|
July 27, 2016
Manganese-Substituted Polyoxometalate as an Effective Shuttle Redox Mediator in Z-Scheme Water Splitting under Visible Light
Kohei Tsuji, Osamu Tomita, Masanobu Higashi, et al.
Organic & Biomolecular Chemistry
|
March 25, 2026
Affinity enhancement of polo-like kinase 1 polo-box domain-binding peptides by <i>N</i>-methylation and lipidation
Kohei Tsuji, Kenan Bai, Xueyuan Huang, et al.
Molecules (Basel, Switzerland)
|
April 25, 2019
Development of Highly Selective 1,2,3-Triazole-containing Peptidic Polo-like Kinase 1 Polo-box Domain-binding Inhibitors
Xue Zhi Zhao, Kohei Tsuji, David Hymel, et al.
Organic & Biomolecular Chemistry
|
February 13, 2025
Diastereoselective synthesis of (<i>Z</i>)-fluoroalkene dipeptide isosteres utilizing chiral auxiliaries
Takuya Kobayakawa, Marisa Arioka, Kenichi Yamamoto, et al.
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Showing results (1-10 of 66) with videos related to
Sort By:
Page
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Yakugaku Zasshi : Journal of the Pharmaceutical Society of Japan
|
October 1, 2025
[Development of Mid-size Bivalent Inhibitors Targeting a Cancer-related Kinase]
Kohei Tsuji
Bioorganic & Medicinal Chemistry
|
July 3, 2024
Design, synthesis and evaluation of bioactivity of peptidomimetics based on chloroalkene dipeptide isosteres
Takuya Kobayakawa, Kohei Tsuji, Hirokazu Tamamura
Bioorganic & Medicinal Chemistry
|
January 7, 2025
Fine-tuning probes for fluorescence polarization binding assays of bivalent ligands against polo-like kinase 1 using full-length protein
Kohei Tsuji, Hirokazu Tamamura, Terrence R Burke
Biological & Pharmaceutical Bulletin
|
July 10, 2024
Application of a Fluorescence Recovery-Based Polo-Like Kinase 1 Binding Assay to Polo-Like Kinase 2 and Polo-Like Kinase 3
Kohei Tsuji, Hirokazu Tamamura, Terrence R Burke
RSC Chemical Biology
|
August 2, 2024
Affinity enhancement of polo-like kinase 1 polo box domain-binding ligands by a bivalent approach using a covalent kinase-binding component
Kohei Tsuji, Hirokazu Tamamura, Terrence R Burke
Analytical Methods : Advancing Methods and Applications
|
September 24, 2020
A new genre of fluorescence recovery assay to evaluate polo-like kinase 1 ATP-competitive inhibitors
Kohei Tsuji, David Hymel, Terrence R Burke
Chemsuschem
|
July 27, 2016
Manganese-Substituted Polyoxometalate as an Effective Shuttle Redox Mediator in Z-Scheme Water Splitting under Visible Light
Kohei Tsuji, Osamu Tomita, Masanobu Higashi, et al.
Organic & Biomolecular Chemistry
|
March 25, 2026
Affinity enhancement of polo-like kinase 1 polo-box domain-binding peptides by <i>N</i>-methylation and lipidation
Kohei Tsuji, Kenan Bai, Xueyuan Huang, et al.
Molecules (Basel, Switzerland)
|
April 25, 2019
Development of Highly Selective 1,2,3-Triazole-containing Peptidic Polo-like Kinase 1 Polo-box Domain-binding Inhibitors
Xue Zhi Zhao, Kohei Tsuji, David Hymel, et al.
Organic & Biomolecular Chemistry
|
February 13, 2025
Diastereoselective synthesis of (<i>Z</i>)-fluoroalkene dipeptide isosteres utilizing chiral auxiliaries
Takuya Kobayakawa, Marisa Arioka, Kenichi Yamamoto, et al.
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