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European Journal of Medicinal Chemistry|May 16, 2006
Novel potent and selective alphavbeta3/alphavbeta5 integrin dual antagonists with reduced binding affinity for human serum albuminPierre Raboisson, Carl L Manthey, Margery Chaikin, et al.Bioorganic & Medicinal Chemistry Letters|May 3, 2005
Non-peptidic alpha(v)beta3 antagonists containing indol-1-yl propionic acidsKristi Leonard, Wenxi Pan, Beth Anaclerio, et al.Bioorganic & Medicinal Chemistry Letters|May 2, 2006
Novel 1,4-benzodiazepine-2,5-diones as Hdm2 antagonists with improved cellular activityKristi Leonard, Juan Jose Marugan, Pierre Raboisson, et al.Bioorganic & Medicinal Chemistry Letters|April 25, 2006
Enantiomerically pure 1,4-benzodiazepine-2,5-diones as Hdm2 antagonistsJuan Jose Marugan, Kristi Leonard, Pierre Raboisson, et al.Journal of Biochemical and Biophysical Methods|December 6, 2005
A functional radioreceptor assay of alpha-V-beta-3 (alphavbeta3) inhibitors in plasma: application as an ex vivo pharmacodynamic modelMargery A Chaikin, Júan José Marugan, Gerald W De Vries, et al.Bioorganic & Medicinal Chemistry Letters|April 11, 2018
Identification and biological evaluation of thiazole-based inverse agonists of RORγtChristian Gege, Maxwell D Cummings, Michael Albers, et al.Bioorganic & Medicinal Chemistry Letters|March 26, 2013
Substituted thieno[2,3-d]pyrimidines as adenosine A2A receptor antagonistsBrian C Shook, Devraj Chakravarty, J Kent Barbay, et al.Bioorganic & Medicinal Chemistry Letters|April 28, 2020
Optimization and biological evaluation of thiazole-bis-amide inverse agonists of RORγtChristian Gege, Michael Albers, Olaf Kinzel, et al.Scientific Reports|December 2, 2016
Pharmacologic modulation of RORγt translates to efficacy in preclinical and translational models of psoriasis and inflammatory arthritisXiaohua Xue, Pejman Soroosh, Aimee De Leon-Tabaldo, et al.Bioorganic & Medicinal Chemistry Letters|April 24, 2019
3-Substituted Quinolines as RORγt Inverse AgonistsVirginia M Tanis, Hariharan Venkatesan, Maxwell D Cummings, et al.Pageof 2