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Drug Discovery Today
|
September 13, 2020
Fragment-based target screening as an empirical approach to prioritising targets: a case study on antibacterials
Peter Canning, Kristian Birchall, Catherine A Kettleborough, et al.
Frontiers in Molecular Neuroscience
|
April 30, 2024
Targeted protein degradation in CNS disorders: a promising route to novel therapeutics?
Sandra Kuemper, Andrew G Cairns, Kristian Birchall, et al.
Journal of Chemical Information and Modeling
|
May 2, 2022
Incorporating Target-Specific Pharmacophoric Information into Deep Generative Models for Fragment Elaboration
Thomas E Hadfield, Fergus Imrie, Andy Merritt, et al.
ACS Chemical Biology
|
October 18, 2014
Competitive binding of a benzimidazole to the histone-binding pocket of the Pygo PHD finger
Thomas C R Miller, Trevor J Rutherford, Kristian Birchall, et al.
ACS Medicinal Chemistry Letters
|
October 15, 2025
Design and Synthesis of Pyrazoline Inhibitors of SARS-CoV‑2 NSP14
Elliott B Smyth, João P Pisco, Kristian Birchall, et al.
BMJ Open
|
June 25, 2013
Antitubercular specific activity of ibuprofen and the other 2-arylpropanoic acids using the HT-SPOTi whole-cell phenotypic assay
Juan D Guzman, Dimitrios Evangelopoulos, Antima Gupta, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 18, 2018
Discovery of potent and selective 5-azaindazole inhibitors of leucine-rich repeat kinase 2 (LRRK2) - Part 1
Joanne Osborne, Kristian Birchall, Denise J Tsagris, et al.
Scientific Reports
|
June 11, 2023
Identification of novel p-cresol inhibitors that reduce Clostridioides difficile's ability to compete with species of the gut microbiome
Mark A Harrison, Rebecca J Farthing, Nyasha Allen, et al.
Journal of Medicinal Chemistry
|
April 3, 2014
Optimization of an imidazopyridazine series of inhibitors of Plasmodium falciparum calcium-dependent protein kinase 1 (PfCDPK1)
Timothy M Chapman, Simon A Osborne, Claire Wallace, et al.
Journal of Medicinal Chemistry
|
April 28, 2018
Design, Synthesis, and Testing of Potent, Selective Hepsin Inhibitors via Application of an Automated Closed-Loop Optimization Platform
Shishir M Pant, Amanda Mukonoweshuro, Bimbisar Desai, et al.
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of 4
Search research articles
Search
Showing results (11-20 of 31) with videos related to
Sort By:
Page
of 4
Drug Discovery Today
|
September 13, 2020
Fragment-based target screening as an empirical approach to prioritising targets: a case study on antibacterials
Peter Canning, Kristian Birchall, Catherine A Kettleborough, et al.
Frontiers in Molecular Neuroscience
|
April 30, 2024
Targeted protein degradation in CNS disorders: a promising route to novel therapeutics?
Sandra Kuemper, Andrew G Cairns, Kristian Birchall, et al.
Journal of Chemical Information and Modeling
|
May 2, 2022
Incorporating Target-Specific Pharmacophoric Information into Deep Generative Models for Fragment Elaboration
Thomas E Hadfield, Fergus Imrie, Andy Merritt, et al.
ACS Chemical Biology
|
October 18, 2014
Competitive binding of a benzimidazole to the histone-binding pocket of the Pygo PHD finger
Thomas C R Miller, Trevor J Rutherford, Kristian Birchall, et al.
ACS Medicinal Chemistry Letters
|
October 15, 2025
Design and Synthesis of Pyrazoline Inhibitors of SARS-CoV‑2 NSP14
Elliott B Smyth, João P Pisco, Kristian Birchall, et al.
BMJ Open
|
June 25, 2013
Antitubercular specific activity of ibuprofen and the other 2-arylpropanoic acids using the HT-SPOTi whole-cell phenotypic assay
Juan D Guzman, Dimitrios Evangelopoulos, Antima Gupta, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 18, 2018
Discovery of potent and selective 5-azaindazole inhibitors of leucine-rich repeat kinase 2 (LRRK2) - Part 1
Joanne Osborne, Kristian Birchall, Denise J Tsagris, et al.
Scientific Reports
|
June 11, 2023
Identification of novel p-cresol inhibitors that reduce Clostridioides difficile's ability to compete with species of the gut microbiome
Mark A Harrison, Rebecca J Farthing, Nyasha Allen, et al.
Journal of Medicinal Chemistry
|
April 3, 2014
Optimization of an imidazopyridazine series of inhibitors of Plasmodium falciparum calcium-dependent protein kinase 1 (PfCDPK1)
Timothy M Chapman, Simon A Osborne, Claire Wallace, et al.
Journal of Medicinal Chemistry
|
April 28, 2018
Design, Synthesis, and Testing of Potent, Selective Hepsin Inhibitors via Application of an Automated Closed-Loop Optimization Platform
Shishir M Pant, Amanda Mukonoweshuro, Bimbisar Desai, et al.
Page
of 4