Showing results (41-50 of 68) with videos related to
Sort By:
Pageof 7
Organic & Biomolecular Chemistry|April 26, 2019
β-Glucuronidase triggers extracellular MMAE release from an integrin-targeted conjugatePaula López Rivas, Christoph Müller, Christian Breunig, et al.Chemmedchem|September 5, 2008
A potent integrin antagonist from a small library of cyclic RGD pentapeptide mimics including benzyl-substituted azabicycloalkane amino acidsDaniela Arosio, Laura Belvisi, Lino Colombo, et al.Chemistry (Weinheim an Der Bergstrasse, Germany)|March 12, 2015
Cyclic isoDGR and RGD peptidomimetics containing bifunctional diketopiperazine scaffolds are integrin antagonistsSilvia Panzeri, Simone Zanella, Daniela Arosio, et al.European Journal of Medicinal Chemistry|July 2, 2013
Modulation of αvβ₃- and α₅β₁-integrin-mediated adhesion by dehydro-β-amino acids containing peptidomimeticsAlessandra Tolomelli, Monica Baiula, Laura Belvisi, et al.RSC Chemical Biology|December 12, 2025
Late-stage peptide modification with salicylaldehyde tag enhances affinity for nuclear factor-kappa B essential modulatorMattia Mason, Kaliroi Peqini, Federico Uggeri, et al.Chemical Communications (Cambridge, England)|February 5, 2015
Designing nanomolar antagonists of DC-SIGN-mediated HIV infection: ligand presentation using molecular rodsStefania Ordanini, Norbert Varga, Vanessa Porkolab, et al.Bioorganic & Medicinal Chemistry|October 11, 2005
Targeting integrins: insights into structure and activity of cyclic RGD pentapeptide mimics containing azabicycloalkane amino acidsLaura Belvisi, Anna Bernardi, Matteo Colombo, et al.Molecules (Basel, Switzerland)|December 19, 2020
Cyclic RGD and <i>iso</i>DGR Integrin Ligands Containing <i>cis</i>-2-amino-1-cyclopentanecarboxylic (<i>cis</i>-β-ACPC) ScaffoldsSilvia Panzeri, Daniela Arosio, Silvia Gazzola, et al.Chemmedchem|March 7, 2019
Synthesis and Biological Evaluation of RGD and isoDGR-Monomethyl Auristatin Conjugates Targeting Integrin α<sub>V</sub> β<sub>3</sub>André Raposo Moreira Dias, Lizeth Bodero, Ana Martins, et al.Journal of Medicinal Chemistry|November 13, 2012
Synthesis and biological evaluation (in vitro and in vivo) of cyclic arginine-glycine-aspartate (RGD) peptidomimetic-paclitaxel conjugates targeting integrin αVβ3Raffaele Colombo, Michele Mingozzi, Laura Belvisi, et al.Pageof 7