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International Journal of Molecular Sciences|January 11, 2024
Mass Spectrometry Study about In Vitro and In Vivo Reaction between Metformin and Glucose: A Preliminary Investigation on Alternative Biological BehaviorGianluca Bartolucci, Marco Pallecchi, Laura Braconi, et al.
Future Microbiology|August 26, 2020
1-benzyl-1,4-diazepane reduces the efflux of resistance-nodulation-cell division pumps in Escherichia coliEnrico Casalone, Tiziano Vignolini, Laura Braconi, et al.
The Journal of Antimicrobial Chemotherapy|November 8, 2021
Characterization of substituted piperazines able to reverse MDR in Escherichia coli strains overexpressing resistance-nodulation-cell division (RND) efflux pumpsEnrico Casalone, Tiziano Vignolini, Laura Braconi, et al.
Molecules (Basel, Switzerland)|January 21, 2022
New Histamine-Related Five-Membered N-Heterocycle Derivatives as Carbonic Anhydrase I ActivatorsNiccolò Chiaramonte, Alessio Gabellini, Andrea Angeli, et al.
Journal of Enzyme Inhibition and Medicinal Chemistry|April 28, 2020
Synthesis and carbonic anhydrase activating properties of a series of 2-amino-imidazolines structurally related to clonidine1Niccolò Chiaramonte, Soumia Maach, Caterina Biliotti, et al.
Molecules (Basel, Switzerland)|April 16, 2020
Dual P-Glycoprotein and CA XII Inhibitors: A New Strategy to Reverse the P-gp Mediated Multidrug Resistance (MDR) in Cancer CellsElisabetta Teodori, Laura Braconi, Silvia Bua, et al.
Bioorganic & Medicinal Chemistry Letters|April 5, 2026
New benzyldiazepane derivatives able to reduce biofilm formation in Escherichia coliLaura Braconi, Elena Perrin, Andrea Carlotta Conti, et al.
Bioorganic Chemistry|August 3, 2019
Sulfonamides incorporating piperazine bioisosteres as potent human carbonic anhydrase I, II, IV and IX inhibitorsNiccolò Chiaramonte, Silvia Bua, Andrea Angeli, et al.
European Journal of Medicinal Chemistry|August 13, 2023
Tetrazole and oxadiazole derivatives as bioisosteres of tariquidar and elacridar: New potent P-gp modulators acting as MDR reversersLaura Braconi, Silvia Dei, Marialessandra Contino, et al.
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