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Journal of Medicinal Chemistry|August 15, 2017
Structure-Affinity Relationships and Structure-Kinetics Relationships of Pyrido[2,1-f]purine-2,4-dione Derivatives as Human Adenosine A3 Receptor AntagonistsLizi Xia, Wessel A C Burger, Jacobus P D van Veldhoven, et al.Journal of Medicinal Chemistry|August 7, 2018
An Affinity-Based Probe for the Human Adenosine A2A ReceptorXue Yang, Thomas J M Michiels, Coen de Jong, et al.Journal of Medicinal Chemistry|July 1, 2015
Structure-Affinity Relationships (SARs) and Structure-Kinetics Relationships (SKRs) of Kv11.1 BlockersZhiyi Yu, Jacobus P D van Veldhoven, Julien Louvel, et al.Expert Opinion on Drug Discovery|October 21, 2015
Mechanistic models enable the rational use of in vitro drug-target binding kinetics for better drug effects in patientsWilhelmus E A de Witte, Yin Cheong Wong, Indira Nederpelt, et al.Journal of Medicinal Chemistry|June 18, 2016
Controlling the Dissociation of Ligands from the Adenosine A2A Receptor through Modulation of Salt Bridge StrengthElena Segala, Dong Guo, Robert K Y Cheng, et al.RSC Medicinal Chemistry|August 4, 2022
Development of subtype-selective covalent ligands for the adenosine A2B receptor by tuning the reactive groupBert L H Beerkens, Xuesong Wang, Maria Avgeropoulou, et al.Journal of the American Chemical Society|July 10, 2026
Automated Parallel Synthesis Accelerates Virtual Screening Hit DiscoverySean M McKenna, Martin Šícho, Cas van der Horst, et al.Bioorganic & Medicinal Chemistry|May 23, 2007
Synthesis and evaluation of homo-bivalent GnRHR ligandsKimberly M Bonger, Richard J B H N van den Berg, Laura H Heitman, et al.Biochemical Pharmacology|April 8, 2022
Kinetic profiling and functional characterization of 8-phenylxanthine derivatives as A2B adenosine receptor antagonistsAnna Vlachodimou, Henk de Vries, Milena Pasoli, et al.Trends in Pharmacological Sciences|December 6, 2017
Structural Mapping of Adenosine Receptor Mutations: Ligand Binding and Signaling MechanismsWillem Jespers, Anke C Schiedel, Laura H Heitman, et al.Pageof 16