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Journal of Medicinal Chemistry|March 25, 2021
Crystal Structure and Subsequent Ligand Design of a Nonriboside Partial Agonist Bound to the Adenosine A2A ReceptorTasia Amelia, Jacobus P D van Veldhoven, Matteo Falsini, et al.Journal of Medicinal Chemistry|February 18, 2021
Design and Characterization of an Intracellular Covalent Ligand for CC Chemokine Receptor 2Natalia V Ortiz Zacarías, Kirti K Chahal, Tereza Šimková, et al.Biochemical Pharmacology|August 7, 2024
CC chemokine receptor 2 is allosterically modulated by sodium ions and amiloride derivatives through a distinct sodium ion binding siteLisa S den Hollander, Annelien J M Zweemer, Olivier J M Béquignon, et al.Journal of Medicinal Chemistry|August 2, 2023
Development of an Affinity-Based Probe to Profile Endogenous Human Adenosine ABert L H Beerkens, Inge M Snijders, Joep Snoeck, et al.Pharmacological Research|November 8, 2025
Kinetic multiplex assay to assess biased signaling of clinical GPCR agonistsJara Bouma, Elisa J M de Koning, Cas van der Horst, et al.Molecular Pharmacology|April 4, 2020
LUF7244 plus Dofetilide Rescues Aberrant Kv11.1 Trafficking and Produces Functional IKv11.1Muge Qile, Yuan Ji, Tyona D Golden, et al.ACS Chemical Biology|August 26, 2024
Labeling of CC Chemokine Receptor 2 with a Versatile Intracellular Allosteric ProbeLisa S den Hollander, Bert L H Beerkens, Sebastian Dekkers, et al.Journal of Medicinal Chemistry|September 14, 2013
Structure-kinetic relationships--an overlooked parameter in hit-to-lead optimization: a case of cyclopentylamines as chemokine receptor 2 antagonistsMaris Vilums, Annelien J M Zweemer, Zhiyi Yu, et al.Journal of Medicinal Chemistry|July 14, 2017
Discovery and Kinetic Profiling of 7-Aryl-1,2,4-triazolo[4,3-a]pyridines: Positive Allosteric Modulators of the Metabotropic Glutamate Receptor 2Maarten L J Doornbos, José María Cid, Jordi Haubrich, et al.European Journal of Medicinal Chemistry|February 11, 2015
When structure-affinity relationships meet structure-kinetics relationships: 3-((Inden-1-yl)amino)-1-isopropyl-cyclopentane-1-carboxamides as CCR2 antagonistsMaris Vilums, Annelien J M Zweemer, Farhana Barmare, et al.Pageof 16