Showing results (141-150 of 160) with videos related to
Sort By:
Pageof 16
Journal of Medicinal Chemistry|September 27, 2018
Pyrrolone Derivatives as Intracellular Allosteric Modulators for Chemokine Receptors: Selective and Dual-Targeting Inhibitors of CC Chemokine Receptors 1 and 2Natalia V Ortiz Zacarías, Jacobus P D van Veldhoven, Laura Portner, et al.RSC Medicinal Chemistry|July 13, 2026
From dual norepinephrine-dopamine reuptake inhibition to selective dopamine reuptake inhibitors: a case of aromatically substituted N,2-cyclopentylaminesMajlen A Dilweg, Willem Jespers, Ameya S Kasture, et al.Scientific Reports|March 2, 2017
A novel CCR2 antagonist inhibits atherogenesis in apoE deficient mice by achieving high receptor occupancyIlze Bot, Natalia V Ortiz Zacarías, Wilhelmus E A de Witte, et al.Proceedings of the National Academy of Sciences of the United States of America|February 20, 2025
The endocannabinoid 2-arachidonoylglycerol is released and transported on demand via extracellular microvesiclesVerena M Straub, Benjamin Barti, Sebastian T Tandar, et al.ACS Chemical Neuroscience|March 13, 2024
Still in Search for an EAAT Activator: GT949 Does Not Activate EAAT2, nor EAAT3 in Impedance and Radioligand Uptake AssaysLieve van Veggel, Tamara A M Mocking, Hubert J Sijben, et al.Nature|December 8, 2016
Structure of CC chemokine receptor 2 with orthosteric and allosteric antagonistsYi Zheng, Ling Qin, Natalia V Ortiz Zacarías, et al.Journal of Medicinal Chemistry|December 11, 2025
Leveraging Targeted Protein Degradation for G Protein-Coupled Receptors: The Development of CCR2 Molecular DegradersKhaled Essa, Natalia V Ortiz Zacarías, Sascha Roth, et al.British Journal of Pharmacology|July 25, 2019
LUF7244, an allosteric modulator/activator of Kv 11.1 channels, counteracts dofetilide-induced torsades de pointes arrhythmia in the chronic atrioventricular block dog modelMuge Qile, Henriette D M Beekman, David J Sprenkeler, et al.Journal of Medicinal Chemistry|July 11, 2024
Highly Selective Drug-Derived Fluorescent Probes for the Cannabinoid Receptor Type 1 (CB1R)Leonard Mach, Anahid Omran, Jara Bouma, et al.Journal of the American Chemical Society|February 9, 2018
Selective Photoaffinity Probe That Enables Assessment of Cannabinoid CB2 Receptor Expression and Ligand Engagement in Human CellsMarjolein Soethoudt, Sara C Stolze, Matthias V Westphal, et al.Pageof 16