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Biochemical Pharmacology|December 13, 2019
Affinity, binding kinetics and functional characterization of draflazine analogues for human equilibrative nucleoside transporter 1 (SLC29A1)Anna Vlachodimou, Konstantina Konstantinopoulou, Adriaan P IJzerman, et al.
Medicinal Research Reviews|April 18, 2024
Pharmacological characterization of allosteric modulators: A case for chemokine receptorsLisa S den Hollander, Adriaan P IJzerman, Laura H Heitman
Purinergic Signalling|December 10, 2015
Scintillation proximity assay (SPA) as a new approach to determine a ligand's kinetic profile. A case in point for the adenosine A1 receptorLizi Xia, Henk de Vries, Ad P IJzerman, et al.
British Journal of Pharmacology|February 14, 2012
Functional efficacy of adenosine A₂A receptor agonists is positively correlated to their receptor residence timeDong Guo, Thea Mulder-Krieger, Adriaan P IJzerman, et al.
Medicinal Research Reviews|February 20, 2014
Drug-target residence time--a case for G protein-coupled receptorsDong Guo, Julia M Hillger, Adriaan P IJzerman, et al.
Methods in Molecular Biology (Clifton, N.J.)|June 2, 2016
Protocol to Study β-Arrestin Recruitment by CB1 and CB2 Cannabinoid ReceptorsMarjolein Soethoudt, Noortje van Gils, Mario van der Stelt, et al.
Drug Discovery Today|August 6, 2017
Label-free technology and patient cells: from early drug development to precision medicineJulia M Hillger, Wai-Ling Lieuw, Laura H Heitman, et al.
Trends in Immunology|April 1, 2014
Bias in chemokine receptor signallingAnnelien J M Zweemer, Jimita Toraskar, Laura H Heitman, et al.
Molecular and Cellular Endocrinology|January 25, 2012
Determination of different putative allosteric binding pockets at the lutropin receptor by using diverse drug-like low molecular weight ligandsLaura H Heitman, Gunnar Kleinau, Johannes Brussee, et al.
ACS Pharmacology & Translational Science|April 17, 2020
Perspective: Implications of Ligand-Receptor Binding Kinetics for Therapeutic Targeting of G Protein-Coupled ReceptorsWijnand J C van der Velden, Laura H Heitman, Mette M Rosenkilde
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