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Biochemical Pharmacology|March 9, 2026
Exploring the binding kinetics of intracellular allosteric antagonists for CC chemokine receptor 2 - a key to improve insurmountable antagonismYao Yao, Lisa S den Hollander, Bente Bleijs, et al.
British Journal of Pharmacology|February 28, 2018
A two-state model for the kinetics of competitive radioligand bindingDong Guo, Lambertus A Peletier, Lloyd Bridge, et al.
British Journal of Pharmacology|July 22, 2014
Molecular mechanism of allosteric modulation at GPCRs: insight from a binding kinetics study at the human A1 adenosine receptorDong Guo, Suzanne N Venhorst, Arnault Massink, et al.
Bioorganic & Medicinal Chemistry|March 14, 2015
Synthesis and biological evaluation of spirocyclic antagonists of CCR2 (chemokine CC receptor subtype 2)Ann Kathrin Strunz, Annelien J M Zweemer, Christina Weiss, et al.
International Journal of Molecular Sciences|April 13, 2024
Computational Characterization of Membrane Proteins as Anticancer Targets: Current Challenges and OpportunitiesMarina Gorostiola González, Pepijn R J Rakers, Willem Jespers, et al.
Biochemical Pharmacology|April 2, 2018
Constitutive activity of the metabotropic glutamate receptor 2 explored with a whole-cell label-free biosensorMaarten L J Doornbos, Ilse Van der Linden, Liesbeth Vereyken, et al.
British Journal of Pharmacology|January 31, 2006
Allosteric modulation, thermodynamics and binding to wild-type and mutant (T277A) adenosine A1 receptors of LUF5831, a novel nonadenosine-like agonistLaura H Heitman, Thea Mulder-Krieger, Ronald F Spanjersberg, et al.
Molecules (Basel, Switzerland)|April 12, 2022
Development of Bicyclo[3.1.0]hexane-Based A3 Receptor Ligands: Closing the Gaps in the Structure-Affinity RelationshipsJan Phillip Lemmerhirt, Andreas Isaak, Rongfang Liu, et al.
Biochemical Pharmacology|November 16, 2023
Dual allosteric and orthosteric pharmacology of synthetic analog cannabidiol-dimethylheptyl, but not cannabidiol, on the cannabinoid CB2 receptorJara Bouma, Jeremy D Broekhuis, Cas van der Horst, et al.
Purinergic Signalling|March 29, 2019
A live cell NanoBRET binding assay allows the study of ligand-binding kinetics to the adenosine A3 receptorMonica Bouzo-Lorenzo, Leigh A Stoddart, Lizi Xia, et al.
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