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Biomedicine & Pharmacotherapy = Biomedecine & Pharmacotherapie|June 10, 2022
Breaking boundaries: Pan BETi disrupt 3D chromatin structure, BD2-selective BETi are strictly epigenetic transcriptional regulatorsLaura M Tsujikawa, Olesya A Kharenko, Stephanie C Stotz, et al.Atherosclerosis|December 1, 2022
Epigenetic BET reader inhibitor apabetalone (RVX-208) counters proinflammatory aortic gene expression in a diet induced obesity mouse model and in human endothelial cellsSylwia Wasiak, Laura M Tsujikawa, Emily Daze, et al.Translational Neuroscience|January 15, 2024
The BET inhibitor apabetalone decreases neuroendothelial proinflammatory activation <i>in vitro</i> and in a mouse model of systemic inflammationSylwia Wasiak, Li Fu, Emily Daze, et al.Clinical Epigenetics|July 14, 2019
Apabetalone (RVX-208) reduces vascular inflammation in vitro and in CVD patients by a BET-dependent epigenetic mechanismLaura M Tsujikawa, Li Fu, Shovon Das, et al.Pageof 2