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Pharmaceutics|February 26, 2022
Identification of a Quinone Derivative as a YAP/TEAD Activity Modulator from a Repurposing LibraryAngela Lauriola, Elisa Uliassi, Matteo Santucci, et al.
European Journal of Medicinal Chemistry|July 18, 2024
Discovery of a new 1-(phenylsulfonyl)-1H-indole derivative targeting the EphA2 receptor with antiproliferative activity on U251 glioblastoma cell lineLorenzo Guidetti, Riccardo Castelli, Alfonso Zappia, et al.
Biochemical Pharmacology|October 5, 2025
Dual targeting of EphAs and KDR axis hampers VEGF-induced angiogenesis and glioma stem cell replicationAlfonso Zappia, Francesca Romana Ferrari, Carmine Giorgio, et al.
Biochemical Pharmacology|February 15, 2026
The rare bile acid isoallolithocholic acid (IALCA) is an EphA2 antagonist sparing FXR and TGR5 receptorsAndrea Blesio, Carmine Giorgio, Francesca Romana Ferrari, et al.
Pharmacological Research|July 5, 2024
Discovery of novel FGF trap small molecules endowed with anti-myeloma activitySara Taranto, Riccardo Castelli, Giuseppe Marseglia, et al.
European Journal of Medicinal Chemistry|December 13, 2025
N-Acylaminoethyltetrahydroquinolines: A new class of melatonin receptor ligands with in vivo activity on glioblastomaAnnalida Bedini, Francesca Galvani, Gian Marco Elisi, et al.
Journal of Medicinal Chemistry|July 17, 2018
Novel Benzazole Derivatives Endowed with Potent Antiheparanase ActivityValentina Noemi Madia, Antonella Messore, Luca Pescatori, et al.
Journal of Medicinal Chemistry|November 13, 2019
Benzisothiazolinone Derivatives as Potent Allosteric Monoacylglycerol Lipase Inhibitors That Functionally Mimic Sulfenylation of Regulatory CysteinesRiccardo Castelli, Laura Scalvini, Federica Vacondio, et al.
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