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ACS Medicinal Chemistry Letters|May 16, 2022
Discovery of 2-Phenylquinolines with Broad-Spectrum Anti-coronavirus ActivityMaria Giulia Nizi, Leentje Persoons, Angela Corona, et al.Nature Genetics|March 9, 2021
Genome-wide CRISPR screening identifies TMEM106B as a proviral host factor for SARS-CoV-2Jim Baggen, Leentje Persoons, Els Vanstreels, et al.Steroids|July 27, 2024
Steroidal 21-imidazolium salt derivatives: Synthesis and anticancer activityNatalia S Sucman, Dmitri Ya Bilan, Sergiu V Cojocari, et al.Journal of Medicinal Chemistry|February 20, 2026
Antiviral Profiling and Cellular Activation of Carbobicyclic Nucleoside AnaloguesStephan Scheeff, Joan Marie Javillo Baguio, Benny Zhibin Liang, et al.Chemmedchem|April 10, 2026
2-Phenylquinolines Exhibit Anti-Severe Acute Respiratory Syndrome Coronavirus-2 Activity Through the Nonstructural Protein 13 Helicase InhibitionGiada Cernicchi, Maria Giulia Nizi, Roberta Emmolo, et al.Cell|July 8, 2023
TMEM106B is a receptor mediating ACE2-independent SARS-CoV-2 cell entryJim Baggen, Maarten Jacquemyn, Leentje Persoons, et al.Plos Pathogens|February 11, 2025
A guanidine-based coronavirus replication inhibitor which targets the nsp15 endoribonuclease and selects for interferon-susceptible mutant virusesBenjamin Van Loy, Eugènia Pujol, Kenichi Kamata, et al.Pageof 7