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Nanoscale|May 20, 2020
Single molecule binding of a ligand to a G-protein-coupled receptor in real time using fluorescence correlation spectroscopy, rendered possible by nano-encapsulation in styrene maleic acid lipid particlesRachael L Grime, Joelle Goulding, Romez Uddin, et al.Journal of Medicinal Chemistry|December 31, 2019
Subtype-Selective Fluorescent Ligands as Pharmacological Research Tools for the Human Adenosine A<sub>2A</sub> ReceptorEleonora Comeo, Nicholas D Kindon, Mark Soave, et al.Journal of Medicinal Chemistry|March 21, 2018
Synthesis and Evaluation of the First Fluorescent Antagonists of the Human P2Y<sub>2</sub> Receptor Based on AR-C118925Sean Conroy, Nicholas D Kindon, Jacqueline Glenn, et al.Organic & Biomolecular Chemistry|July 25, 2013
Conversion of a non-selective adenosine receptor antagonist into A3-selective high affinity fluorescent probes using peptide-based linkersAndrea J Vernall, Leigh A Stoddart, Stephen J Briddon, et al.Journal of Medicinal Chemistry|June 23, 2022
Optimization of Peptide Linker-Based Fluorescent Ligands for the Histamine H<sub>1</sub> ReceptorZhi Yuan Kok, Leigh A Stoddart, Sarah J Mistry, et al.Journal of Medicinal Chemistry|March 21, 2023
Small-Molecule Fluorescent Ligands for the CXCR4 Chemokine ReceptorSebastian Dekkers, Birgit Caspar, Joëlle Goulding, et al.Nature Methods|June 2, 2015
Application of BRET to monitor ligand binding to GPCRsLeigh A Stoddart, Elizabeth K M Johnstone, Amanda J Wheal, et al.Communications Biology|November 28, 2020
Ligand-directed covalent labelling of a GPCR with a fluorescent tag in live cellsLeigh A Stoddart, Nicholas D Kindon, Omolade Otun, et al.Molecular Pharmacology|April 19, 2011
Extracellular loop 2 of the free fatty acid receptor 2 mediates allosterism of a phenylacetamide ago-allosteric modulatorNicola J Smith, Richard J Ward, Leigh A Stoddart, et al.Scientific Reports|January 27, 2018
Development of novel fluorescent histamine H<sub>1</sub>-receptor antagonists to study ligand-binding kinetics in living cellsLeigh A Stoddart, Andrea J Vernall, Monica Bouzo-Lorenzo, et al.Pageof 5