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Expert Opinion on Therapeutic Patents|March 24, 2020
GABAA receptor subtype modulators in medicinal chemistry: an updated patent review (2014-present)Letizia Crocetti, Gabriella GuerriniBioorganic & Medicinal Chemistry|May 25, 2025
Recent breakthroughs in synthetic small molecules targeting SARS-CoV-2 Mpro from 2022 to 2024Laura Braconi, Alice Sosic, Letizia CrocettiMolecules (Basel, Switzerland)|August 12, 2022
An Overview of PDE4 Inhibitors in Clinical Trials: 2010 to Early 2022Letizia Crocetti, Giuseppe Floresta, Agostino Cilibrizzi, et al.International Journal of Molecular Sciences|July 29, 2023
PDE4 Inhibitors: Profiling Hits through the Multitude of Structural ClassesJian Jin, Francesca Mazzacuva, Letizia Crocetti, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|May 6, 2020
Repurposing strategies on pyridazinone-based series by pharmacophore- and structure-driven screeningGiuseppe Floresta, Letizia Crocetti, Maria Paola Giovannoni, et al.Molecules (Basel, Switzerland)|April 13, 2023
4,5-Dihydro-5-Oxo-Pyrazolo[1,5-a]Thieno[2,3-c]Pyrimidine: A Novel Scaffold Containing Thiophene Ring. Chemical Reactivity and In Silico Studies to Predict the Profile to GABAA Receptor SubtypeLetizia Crocetti, Gabriella Guerrini, Fabrizio Melani, et al.International Journal of Molecular Sciences|October 16, 2024
3,8-Disubstituted Pyrazolo[1,5-a]quinazoline as GABAA Receptor Modulators: Synthesis, Electrophysiological Assays, and Molecular Modelling StudiesLetizia Crocetti, Gabriella Guerrini, Fabrizio Melani, et al.Molecules (Basel, Switzerland)|March 29, 2023
Steered Molecular Dynamics Simulations Study on FABP4 InhibitorsRosario Tomarchio, Vincenzo Patamia, Chiara Zagni, et al.International Journal of Molecular Sciences|November 11, 2022
GABAA Receptor Modulators with a Pyrazolo[1,5-a]quinazoline Core: Synthesis, Molecular Modelling Studies and Electrophysiological AssaysLetizia Crocetti, Gabriella Guerrini, Fabrizio Melani, et al.Mini Reviews in Medicinal Chemistry|June 14, 2016
α2 Adrenoceptor: a Target for Neuropathic Pain TreatmentLorenzo Di Cesare Mannelli, Laura Micheli, Letizia Crocetti, et al.Pageof 6