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Bioorganic & Medicinal Chemistry Letters|December 28, 2020
'Proximity frequencies' a new parameter to evaluate the profile of GABAAR modulatorsLetizia Crocetti, Gabriella Guerrini, Niccolò Cantini, et al.
Bioorganic & Medicinal Chemistry Letters|February 3, 2009
A thiabendazole sulfonamide shows potent inhibitory activity against mammalian and nematode alpha-carbonic anhydrasesLetizia Crocetti, Alfonso Maresca, Claudia Temperini, et al.
International Journal of Molecular Sciences|March 24, 2019
Synthesis of New GABAA Receptor Modulator with Pyrazolo[1,5-a]quinazoline (PQ) ScaffoldGabriella Guerrini, Claudia Vergelli, Niccolò Cantini, et al.
Molecules (Basel, Switzerland)|June 19, 2024
Anti-Inflammatory Activity of Pyrazolo[1,5-a]quinazolinesLetizia Crocetti, Andrei I Khlebnikov, Gabriella Guerrini, et al.
Frontiers in Chemistry|October 9, 2020
Novel Sulfonamide Analogs of Sivelestat as Potent Human Neutrophil Elastase InhibitorsLetizia Crocetti, Maria Paola Giovannoni, Niccolò Cantini, et al.
Journal of Enzyme Inhibition and Medicinal Chemistry|January 2, 2026
Insights into the complexity of SARS-CoV-2 Mpro inhibition: Ebselen and its derivatives impair dimerisation of the enzymeSimone Fabbian, Silvia Fabi, Laurin Schwarz, et al.
Acta Chimica Slovenica|September 25, 2013
New Pyrazolo[1',5':1,6]pyrimido[4,5-d]pyridazin-4(3H)-ones Fluoroderivatives as Human A1 Adenosine Receptor LigandsAlessia Graziano, Maria Paola Giovannoni, Agostino Cilibrizzi, et al.
European Journal of Medicinal Chemistry|June 26, 2021
Design and synthesis of the first indole-based blockers of Panx-1 channelLetizia Crocetti, Gabriella Guerrini, Sara Puglioli, et al.
Archiv Der Pharmazie|July 30, 2023
Optimization of 4-amino-pyridazin-3(2H)-one as a valid core scaffold for FABP4 inhibitorsGiuseppe Floresta, Letizia Crocetti, Renan Rodrigues de Oliveira Silva, et al.
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