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Bioorganic & Medicinal Chemistry|July 12, 2011
Design, synthesis and evaluation of N-benzoylindazole derivatives and analogues as inhibitors of human neutrophil elastaseLetizia Crocetti, Maria Paola Giovannoni, Igor A Schepetkin, et al.International Journal of Molecular Sciences|May 14, 2022
New Panx-1 Blockers: Synthesis, Biological Evaluation and Molecular Dynamic StudiesLetizia Crocetti, Gabriella Guerrini, Maria Paola Giovannoni, et al.International Journal of Molecular Sciences|February 11, 2023
Design, Synthesis and Pharmacological Evaluation of New Quinoline-Based Panx-1 Channel BlockersLetizia Crocetti, Maria Paola Giovannoni, Gabriella Guerrini, et al.Journal of Medicinal Chemistry|November 11, 2017
Identification of a New Pyrazolo[1,5-a]quinazoline Ligand Highly Affine to γ-Aminobutyric Type A (GABAA) Receptor Subtype with Anxiolytic-Like and Antihyperalgesic ActivityGabriella Guerrini, Giovanna Ciciani, Letizia Crocetti, et al.Bioorganic & Medicinal Chemistry|November 3, 2018
1H-pyrrolo[2,3-b]pyridine: A new scaffold for human neutrophil elastase (HNE) inhibitorsLetizia Crocetti, Maria Paola Giovannoni, Igor A Schepetkin, et al.Purinergic Signalling|January 20, 2026
Abnormal purinergic signaling contributes to development of renal cysts in autosomal dominant polycystic kidney diseaseVeniamin Ivanov, Andrew Wu, Letizia Crocetti, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|June 15, 2017
Isoxazol-5(2H)-one: a new scaffold for potent human neutrophil elastase (HNE) inhibitorsClaudia Vergelli, Igor A Schepetkin, Letizia Crocetti, et al.Bioorganic & Medicinal Chemistry|November 21, 2020
Exploration of nitrogen heterocycle scaffolds for the development of potent human neutrophil elastase inhibitorsNiccolò Cantini, Andrei I Khlebnikov, Letizia Crocetti, et al.Bioorganic & Medicinal Chemistry|May 22, 2012
Synthesis, enantioresolution, and activity profile of chiral 6-methyl-2,4-disubstituted pyridazin-3(2H)-ones as potent N-formyl peptide receptor agonistsAgostino Cilibrizzi, Igor A Schepetkin, Gianluca Bartolucci, et al.Drug Development Research|July 31, 2016
Synthesis and Pharmacological Evaluation of Indole Derivatives as Deaza Analogues of Potent Human Neutrophil Elastase InhibitorsLetizia Crocetti, Igor A Schepetkin, Giovanna Ciciani, et al.Pageof 6