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Medicinal Research Reviews|April 18, 2024
Pharmacological characterization of allosteric modulators: A case for chemokine receptorsLisa S den Hollander, Adriaan P IJzerman, Laura H HeitmanBiochemical Pharmacology|March 9, 2026
Exploring the binding kinetics of intracellular allosteric antagonists for CC chemokine receptor 2 - a key to improve insurmountable antagonismYao Yao, Lisa S den Hollander, Bente Bleijs, et al.Journal of Medicinal Chemistry|November 20, 2019
Synthesis and Pharmacological Evaluation of Triazolopyrimidinone Derivatives as Noncompetitive, Intracellular Antagonists for CC Chemokine Receptors 2 and 5Natalia V Ortiz Zacarías, Jacobus P D van Veldhoven, Lisa S den Hollander, et al.Biochemical Pharmacology|August 7, 2024
CC chemokine receptor 2 is allosterically modulated by sodium ions and amiloride derivatives through a distinct sodium ion binding siteLisa S den Hollander, Annelien J M Zweemer, Olivier J M Béquignon, et al.ACS Chemical Biology|August 26, 2024
Labeling of CC Chemokine Receptor 2 with a Versatile Intracellular Allosteric ProbeLisa S den Hollander, Bert L H Beerkens, Sebastian Dekkers, et al.Pageof 1