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Journal of Enzyme Inhibition and Medicinal Chemistry|August 27, 2020
Efficient synthesis, biological evaluation, and docking study of isatin based derivatives as caspase inhibitorsLoghman Firoozpour, Lixin Gao, Setareh Moghimi, et al.European Journal of Medicinal Chemistry|September 9, 2025
Discovery of 2-tetrahydroisoquinoline substituted quinazoline derivatives as lysine methyltransferase G9a inhibitors with in vivo antitumor efficacyMengjie Shao, Lixin Gao, Jiahui Xu, et al.ACS Medicinal Chemistry Letters|August 14, 2024
Design, Synthesis, and Biological Evaluation of 2,4-Diaminopyrimidine Derivatives as Potent CDK7 InhibitorsHualin Zhang, Yutong Tu, Zhaofan Tao, et al.Archiv Der Pharmazie|November 22, 2025
Identification of Novel β-Lactam Derivatives as Proteasome Inhibitors for Antitumor TherapyYu Cao, Gaoya Xu, Lixin Gao, et al.RSC Medicinal Chemistry|May 4, 2026
Beyond acrylamide: a structure-guided investigation of covalent warheads in the development of CDK7 inhibitorsYu Cao, Yiqing Huang, Yunlong Pan, et al.Journal of Medicinal Chemistry|July 9, 2026
Discovery of Novel Isoxazole-Based FXR Agonists Containing a 1,2,4-Oxadiazol-5(4H)-one RingMingliang Liu, Jingjing Shi, Yi Zang, et al.Journal of Medicinal Chemistry|September 29, 2018
Development of Macrocyclic Peptides Containing Epoxyketone with Oral Availability as Proteasome InhibitorsDaqiang Li, Xiaotuan Zhang, Xiaodong Ma, et al.Journal of Medicinal Chemistry|November 17, 2022
Discovery of Novel N-(5-(Pyridin-3-yl)-1H-indazol-3-yl)benzamide Derivatives as Potent Cyclin-Dependent Kinase 7 Inhibitors for the Treatment of Autosomal Dominant Polycystic Kidney DiseaseBowen Yang, Haoran Zhang, Na Li, et al.European Journal of Medicinal Chemistry|February 26, 2022
Metabolism guided optimization of peptidomimetics as non-covalent proteasome inhibitors for cancer treatmentYu Cao, Yutong Tu, Liping Fu, et al.Small (Weinheim an Der Bergstrasse, Germany)|February 21, 2025
pH-Responsive DNA-Functionalized Liquid Metal-Organic Frameworks (L-MOFs) as Molecular Sponges for Ultrasensitive and Label-Free SERS Detection of Folic AcidXu Liu, Liliia Glazutdinova, Guangrun Wu, et al.Pageof 7