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Journal of Medicinal Chemistry
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June 17, 2008
Discovery of a potent, selective, and orally bioavailable c-Met inhibitor: 1-(2-hydroxy-2-methylpropyl)-N-(5-(7-methoxyquinolin-4-yloxy)pyridin-2-yl)-5-methyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazole-4-carboxamide (AMG 458)
Longbin Liu, Aaron Siegmund, Ning Xi, et al.
Bioorganic & Medicinal Chemistry Letters
|
July 27, 2012
Synthesis and structure-activity relationships of dual PI3K/mTOR inhibitors based on a 4-amino-6-methyl-1,3,5-triazine sulfonamide scaffold
Ryan P Wurz, Longbin Liu, Kevin Yang, et al.
Journal of Medicinal Chemistry
|
March 12, 2014
Small molecule disruptors of the glucokinase-glucokinase regulatory protein interaction: 3. Structure-activity relationships within the aryl carbinol region of the N-arylsulfonamido-N'-arylpiperazine series
Nobuko Nishimura, Mark H Norman, Longbin Liu, et al.
Journal of Medicinal Chemistry
|
May 27, 2011
Phospshoinositide 3-kinase (PI3K)/mammalian target of rapamycin (mTOR) dual inhibitors: discovery and structure-activity relationships of a series of quinoline and quinoxaline derivatives
Nobuko Nishimura, Aaron Siegmund, Longbin Liu, et al.
Journal of Medicinal Chemistry
|
September 4, 2008
Design, synthesis, and biological evaluation of potent c-Met inhibitors
Noel D D'Angelo, Steven F Bellon, Shon K Booker, et al.
Science Translational Medicine
|
February 2, 2022
Development of a ligand for in vivo imaging of mutant huntingtin in Huntington's disease
Daniele Bertoglio, Jonathan Bard, Manuela Hessmann, et al.
Scientific Reports
|
September 10, 2021
Pharmacological characterization of mutant huntingtin aggregate-directed PET imaging tracer candidates
Frank Herrmann, Manuela Hessmann, Sabine Schaertl, et al.
Journal of Medicinal Chemistry
|
February 22, 2011
Discovery and optimization of a series of benzothiazole phosphoinositide 3-kinase (PI3K)/mammalian target of rapamycin (mTOR) dual inhibitors
Noel D D'Angelo, Tae-Seong Kim, Kristin Andrews, et al.
Journal of Medicinal Chemistry
|
January 11, 2014
Small molecule disruptors of the glucokinase-glucokinase regulatory protein interaction: 2. Leveraging structure-based drug design to identify analogues with improved pharmacokinetic profiles
David J St Jean, Kate S Ashton, Michael D Bartberger, et al.
Frontiers in Pharmacology
|
March 7, 2019
Drug Repurposing: The Anthelmintics Niclosamide and Nitazoxanide Are Potent TMEM16A Antagonists That Fully Bronchodilate Airways
Kent Miner, Katja Labitzke, Benxian Liu, et al.
Page
of 6
Search research articles
Search
Showing results (41-50 of 60) with videos related to
Sort By:
Page
of 6
Journal of Medicinal Chemistry
|
June 17, 2008
Discovery of a potent, selective, and orally bioavailable c-Met inhibitor: 1-(2-hydroxy-2-methylpropyl)-N-(5-(7-methoxyquinolin-4-yloxy)pyridin-2-yl)-5-methyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazole-4-carboxamide (AMG 458)
Longbin Liu, Aaron Siegmund, Ning Xi, et al.
Bioorganic & Medicinal Chemistry Letters
|
July 27, 2012
Synthesis and structure-activity relationships of dual PI3K/mTOR inhibitors based on a 4-amino-6-methyl-1,3,5-triazine sulfonamide scaffold
Ryan P Wurz, Longbin Liu, Kevin Yang, et al.
Journal of Medicinal Chemistry
|
March 12, 2014
Small molecule disruptors of the glucokinase-glucokinase regulatory protein interaction: 3. Structure-activity relationships within the aryl carbinol region of the N-arylsulfonamido-N'-arylpiperazine series
Nobuko Nishimura, Mark H Norman, Longbin Liu, et al.
Journal of Medicinal Chemistry
|
May 27, 2011
Phospshoinositide 3-kinase (PI3K)/mammalian target of rapamycin (mTOR) dual inhibitors: discovery and structure-activity relationships of a series of quinoline and quinoxaline derivatives
Nobuko Nishimura, Aaron Siegmund, Longbin Liu, et al.
Journal of Medicinal Chemistry
|
September 4, 2008
Design, synthesis, and biological evaluation of potent c-Met inhibitors
Noel D D'Angelo, Steven F Bellon, Shon K Booker, et al.
Science Translational Medicine
|
February 2, 2022
Development of a ligand for in vivo imaging of mutant huntingtin in Huntington's disease
Daniele Bertoglio, Jonathan Bard, Manuela Hessmann, et al.
Scientific Reports
|
September 10, 2021
Pharmacological characterization of mutant huntingtin aggregate-directed PET imaging tracer candidates
Frank Herrmann, Manuela Hessmann, Sabine Schaertl, et al.
Journal of Medicinal Chemistry
|
February 22, 2011
Discovery and optimization of a series of benzothiazole phosphoinositide 3-kinase (PI3K)/mammalian target of rapamycin (mTOR) dual inhibitors
Noel D D'Angelo, Tae-Seong Kim, Kristin Andrews, et al.
Journal of Medicinal Chemistry
|
January 11, 2014
Small molecule disruptors of the glucokinase-glucokinase regulatory protein interaction: 2. Leveraging structure-based drug design to identify analogues with improved pharmacokinetic profiles
David J St Jean, Kate S Ashton, Michael D Bartberger, et al.
Frontiers in Pharmacology
|
March 7, 2019
Drug Repurposing: The Anthelmintics Niclosamide and Nitazoxanide Are Potent TMEM16A Antagonists That Fully Bronchodilate Airways
Kent Miner, Katja Labitzke, Benxian Liu, et al.
Page
of 6