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Future Medicinal Chemistry|November 23, 2016
Modern tools for the chemical ligation and synthesis of modified peptides and proteinsLuca Gentilucci, Pierluigi Tosi, Adriano Bauer, et al.Amino Acids|May 5, 2011
A straightforward route to enantiopure 2-substituted-3,4-dehydro-β-proline via ring closing metathesisAlessandra Tolomelli, Luca Gentilucci, Elisa Mosconi, et al.Biomedicines|February 24, 2024
Conjecturing about Small-Molecule Agonists and Antagonists of α4β1 Integrin: From Mechanistic Insight to Potential Therapeutic ApplicationsTingting He, Daria Giacomini, Alessandra Tolomelli, et al.Molecules (Basel, Switzerland)|October 27, 2022
PacDOCK: A Web Server for Positional Distance-Based and Interaction-Based Analysis of Docking ResultsJacopo Carbone, Alessia Ghidini, Antonio Romano, et al.Medicinal Chemistry (Shariqah (United Arab Emirates))|July 20, 2006
A novel family of minimal PMRI cyclic peptides as versatile scaffolds for generating new molecular topologyLuca Gentilucci, Giuliana Cardillo, Alessandra Tolomelli, et al.Biomedicines|March 28, 2026
Computational Pharmacodynamic Analysis of Cyclopeptides Derived from c[Trp-Phe-D-Pro-Phe] (CJ-15,208), an Unusual Class of Mixed μ/k-Opioid Receptor Ligands Lacking the Traditional PharmacophoresMarco Francescato, Hang Liao, Lorenzo Cavina, et al.Organic Letters|May 20, 2008
Synthesis of dehydro-beta-amino esters via highly regioselective amination of allylic carbonatesFides Benfatti, Giuliana Cardillo, Luca Gentilucci, et al.Organic & Biomolecular Chemistry|February 10, 2012
Expedient synthesis of pseudo-Pro-containing peptides: towards constrained peptidomimetics and foldamersRossella De Marco, Alessandra Tolomelli, Marilena Campitiello, et al.Journal of Medicinal Chemistry|May 31, 2002
Endomorphin-1 analogues containing beta-proline are mu-opioid receptor agonists and display enhanced enzymatic hydrolysis resistanceGiuliana Cardillo, Luca Gentilucci, Ahmed R Qasem, et al.Journal of Medicinal Chemistry|September 22, 2012
Opioid activity profiles of oversimplified peptides lacking in the protonable N-terminusRossella De Marco, Alessandra Tolomelli, Santi Spampinato, et al.Pageof 8