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Mini Reviews in Medicinal Chemistry|July 3, 2013
Activin Receptor-like kinase 1: a novel anti-angiogenesis target from TGF-β familyLuca Vecchia, Carla Olivieri, Claudia ScottiCurrent Opinion in Structural Biology|July 11, 2024
Pioneer factors: Emerging rules of engagement for transcription factors on chromatinized DNAManuel Carminati, Luca Vecchia, Lisa Stoos, et al.Journal of Immunotherapy (Hagerstown, Md. : 1997)|October 13, 2011
Targeted drug delivery using immunoconjugates: principles and applicationsMaria Valentina Pasquetto, Luca Vecchia, Daniele Covini, et al.Nature|July 24, 2020
Glypicans shield the Wnt lipid moiety to enable signalling at a distanceIan J McGough, Luca Vecchia, Benjamin Bishop, et al.Medchemcomm|September 20, 2019
Discovery of 2-phenoxyacetamides as inhibitors of the Wnt-depalmitoleating enzyme NOTUM from an X-ray fragment screenBenjamin N Atkinson, David Steadman, Yuguang Zhao, et al.Molecular Cell|February 12, 2026
The human BAF chromatin remodeler processes nucleosomes bound by pioneer transcription factors OCT4-SOX2Joscha Weiss, Luca Vecchia, David Domjan, et al.Journal of Medicinal Chemistry|October 30, 2020
5-Phenyl-1,3,4-oxadiazol-2(3<i>H</i>)-ones Are Potent Inhibitors of Notum Carboxylesterase Activity Identified by the Optimization of a Crystallographic Fragment Screening HitWilliam Mahy, Nicky J Willis, Yuguang Zhao, et al.Journal of Medicinal Chemistry|August 14, 2020
Screening of a Custom-Designed Acid Fragment Library Identifies 1-Phenylpyrroles and 1-Phenylpyrrolidines as Inhibitors of Notum Carboxylesterase ActivityWilliam Mahy, Mikesh Patel, David Steadman, et al.ACS Chemical Neuroscience|June 22, 2022
Structural Analysis and Development of Notum Fragment Screening HitsYuguang Zhao, William Mahy, Nicky J Willis, et al.Journal of Medicinal Chemistry|May 10, 2022
Design of a Potent, Selective, and Brain-Penetrant Inhibitor of Wnt-Deactivating Enzyme Notum by Optimization of a Crystallographic Fragment HitNicky J Willis, William Mahy, James Sipthorp, et al.Pageof 2