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ACS Omega|February 16, 2026
Big Data for Drug Discovery: Some Historical Landscape, Considerations, and Applications for a Medicinal ChemistJoão A L de Lima, Lucas Silva Franco, Lídia M LimaPharmaceuticals (Basel, Switzerland)|August 26, 2023
The Magic Methyl and Its Tricks in Drug Discovery and DevelopmentPedro de Sena Murteira Pinheiro, Lucas Silva Franco, Carlos Alberto Manssour FragaRSC Advances|February 23, 2024
Stereochemical insights into β-amino-N-acylhydrazones and their impact on DPP-4 inhibitionEduardo Reina, Lucas Silva Franco, Teiliane Rodrigues Carneiro, et al.Expert Opinion on Drug Discovery|March 8, 2024
Molecular hybridization: a powerful tool for multitarget drug discoveryPedro de Sena Murteira Pinheiro, Lucas Silva Franco, Tadeu Lima Montagnoli, et al.Pharmaceuticals (Basel, Switzerland)|June 27, 2024
Remapping the Chemical Space and the Pharmacological Space of Drugs: What Can We Expect from the Road Ahead?Lucas Silva Franco, Bárbara da Silva Mascarenhas de Jesus, Pedro de Sena Murteira Pinheiro, et al.Molecules (Basel, Switzerland)|January 8, 2025
Regioselective Nucleophilic Aromatic Substitution: Theoretical and Experimental Insights into 4-Aminoquinazoline Synthesis as a Privileged Structure in Medicinal ChemistryMaria Letícia de Castro Barbosa, Pedro de Sena Murteira Pinheiro, Raissa Alves da Conceição, et al.ACS Omega|July 14, 2025
Drug Repurposing by Virtual Screening: Identification of New Already Approved ROCK Inhibitors as Promising Drugs to Target NeurodegenerationLucas Silva Franco, Daniel Alencar Rodrigues, Gabriela Joras Baumart, et al.Pharmaceuticals (Basel, Switzerland)|June 26, 2026
Multitarget Strategy for Treatment of Pulmonary Arterial Hypertension: Combination of Mesenchymal Cells with Novel PDE-4 InhibitorBruno Eduardo Dematté, Juliana Ferreira Vasques, Almir Jordão da Silva-Junior, et al.Pharmaceuticals (Basel, Switzerland)|July 27, 2022
Discovery of Putative Dual Inhibitor of Tubulin and EGFR by Phenotypic Approach on LASSBio-1586 HomologsGisele Barbosa, Luis Gabriel Valdivieso Gelves, Caroline Marques Xavier Costa, et al.ACS Bio & Med Chem Au|April 20, 2026
Discovery of N‑Acylhydrazone Derivatives as ROCK Inhibitors: A Journey from Virtual Screening and Structure-Based De Novo Design to the Identification of ROCK2 Selective Inhibitors and BeyondPedro de Sena Murteira Pinheiro, Lucas Silva Franco, Raysa Magali Pillpe-Meza, et al.Pageof 2