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Luscombe

Showing results (651-660 of 713) with videos related to

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Journal of Chemical Information and Modeling|September 30, 2010
Lead optimization using matched molecular pairs: inclusion of contextual information for enhanced prediction of HERG inhibition, solubility, and lipophilicityGeorge Papadatos, Muhammad Alkarouri, Valerie J Gillet, et al.
Bioorganic & Medicinal Chemistry Letters|December 25, 2018
Novel M<sub>4</sub> positive allosteric modulators derived from questioning the role and impact of a presumed intramolecular hydrogen-bonding motif in β-amino carboxamide-harboring ligandsMichael S Poslusney, James M Salovich, Michael R Wood, et al.
Bioorganic & Medicinal Chemistry Letters|June 22, 2017
Discovery and optimization of 3-(4-aryl/heteroarylsulfonyl)piperazin-1-yl)-6-(piperidin-1-yl)pyridazines as novel, CNS penetrant pan-muscarinic antagonistsAaron M Bender, Rebecca L Weiner, Vincent B Luscombe, et al.
Bioorganic & Medicinal Chemistry Letters|September 4, 2017
Discovery of a novel, CNS penetrant M<sub>4</sub> PAM chemotype based on a 6-fluoro-4-(piperidin-1-yl)quinoline-3-carbonitrile coreBlake R Bewley, Paul K Spearing, Rebecca L Weiner, et al.
Epigenetics|March 2, 2016
Quantitative genome-wide methylation analysis of high-grade non-muscle invasive bladder cancerMark O Kitchen, Richard T Bryan, Richard D Emes, et al.
Bioorganic & Medicinal Chemistry Letters|October 18, 2017
Discovery of a novel 2,4-dimethylquinoline-6-carboxamide M<sub>4</sub> positive allosteric modulator (PAM) chemotype via scaffold hoppingMadeline F Long, Julie L Engers, Sichen Chang, et al.
Genome Research|April 10, 2010
Multiplexed massively parallel SELEX for characterization of human transcription factor binding specificitiesArttu Jolma, Teemu Kivioja, Jarkko Toivonen, et al.
Ebiomedicine|June 23, 2016
Intra-Tumor Genetic Heterogeneity in Wilms Tumor: Clonal Evolution and Clinical ImplicationsGeorge D Cresswell, John R Apps, Tasnim Chagtai, et al.
Bioorganic & Medicinal Chemistry Letters|December 1, 2019
Discovery of a novel 2,3-dimethylimidazo[1,2-a]pyrazine-6-carboxamide M<sub>4</sub> positive allosteric modulator (PAM) chemotypeKayla J Temple, Julie L Engers, Madeline F Long, et al.
Nature|January 25, 2023
Annelid functional genomics reveal the origins of bilaterian life cyclesFrancisco M Martín-Zamora, Yan Liang, Kero Guynes, et al.
Pageof 72

Showing results (651-660 of 713) with videos related to

Sort By:
Pageof 72
Journal of Chemical Information and Modeling|September 30, 2010
Lead optimization using matched molecular pairs: inclusion of contextual information for enhanced prediction of HERG inhibition, solubility, and lipophilicityGeorge Papadatos, Muhammad Alkarouri, Valerie J Gillet, et al.
Bioorganic & Medicinal Chemistry Letters|December 25, 2018
Novel M<sub>4</sub> positive allosteric modulators derived from questioning the role and impact of a presumed intramolecular hydrogen-bonding motif in β-amino carboxamide-harboring ligandsMichael S Poslusney, James M Salovich, Michael R Wood, et al.
Bioorganic & Medicinal Chemistry Letters|June 22, 2017
Discovery and optimization of 3-(4-aryl/heteroarylsulfonyl)piperazin-1-yl)-6-(piperidin-1-yl)pyridazines as novel, CNS penetrant pan-muscarinic antagonistsAaron M Bender, Rebecca L Weiner, Vincent B Luscombe, et al.
Bioorganic & Medicinal Chemistry Letters|September 4, 2017
Discovery of a novel, CNS penetrant M<sub>4</sub> PAM chemotype based on a 6-fluoro-4-(piperidin-1-yl)quinoline-3-carbonitrile coreBlake R Bewley, Paul K Spearing, Rebecca L Weiner, et al.
Epigenetics|March 2, 2016
Quantitative genome-wide methylation analysis of high-grade non-muscle invasive bladder cancerMark O Kitchen, Richard T Bryan, Richard D Emes, et al.
Bioorganic & Medicinal Chemistry Letters|October 18, 2017
Discovery of a novel 2,4-dimethylquinoline-6-carboxamide M<sub>4</sub> positive allosteric modulator (PAM) chemotype via scaffold hoppingMadeline F Long, Julie L Engers, Sichen Chang, et al.
Genome Research|April 10, 2010
Multiplexed massively parallel SELEX for characterization of human transcription factor binding specificitiesArttu Jolma, Teemu Kivioja, Jarkko Toivonen, et al.
Ebiomedicine|June 23, 2016
Intra-Tumor Genetic Heterogeneity in Wilms Tumor: Clonal Evolution and Clinical ImplicationsGeorge D Cresswell, John R Apps, Tasnim Chagtai, et al.
Bioorganic & Medicinal Chemistry Letters|December 1, 2019
Discovery of a novel 2,3-dimethylimidazo[1,2-a]pyrazine-6-carboxamide M<sub>4</sub> positive allosteric modulator (PAM) chemotypeKayla J Temple, Julie L Engers, Madeline F Long, et al.
Nature|January 25, 2023
Annelid functional genomics reveal the origins of bilaterian life cyclesFrancisco M Martín-Zamora, Yan Liang, Kero Guynes, et al.
Pageof 72