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Molecular Cancer Therapeutics
|
August 14, 2021
Clinical Positioning of the IAP Antagonist Tolinapant (ASTX660) in Colorectal Cancer
Nyree Crawford, Katie J Stott, Tamas Sessler, et al.
Molecular Cancer Therapeutics
|
May 12, 2012
Chemosensitization of cancer cells by KU-0060648, a dual inhibitor of DNA-PK and PI-3K
Joanne M Munck, Michael A Batey, Yan Zhao, et al.
ACS Medicinal Chemistry Letters
|
July 21, 2015
Fragment-Based Discovery of Potent and Selective DDR1/2 Inhibitors
Christopher W Murray, Valerio Berdini, Ildiko M Buck, et al.
Journal of Medicinal Chemistry
|
August 10, 2018
A Fragment-Derived Clinical Candidate for Antagonism of X-Linked and Cellular Inhibitor of Apoptosis Proteins: 1-(6-[(4-Fluorophenyl)methyl]-5-(hydroxymethyl)-3,3-dimethyl-1 H,2 H,3 H-pyrrolo[3,2- b]pyridin-1-yl)-2-[(2 R,5 R)-5-methyl-2-([(3R)-3-methylmorpholin-4-yl]methyl)piperazin-1-yl]ethan-1-one (ASTX660)
Christopher N Johnson, Jong Sook Ahn, Ildiko M Buck, et al.
The Journal of Clinical Investigation
|
October 4, 2019
Selective DNA-PKcs inhibition extends the therapeutic index of localized radiotherapy and chemotherapy
Catherine E Willoughby, Yanyan Jiang, Huw D Thomas, et al.
Molecular Cancer Therapeutics
|
July 31, 2021
ASTX029, a Novel Dual-mechanism ERK Inhibitor, Modulates Both the Phosphorylation and Catalytic Activity of ERK
Joanne M Munck, Valerio Berdini, Luke Bevan, et al.
Journal of Medicinal Chemistry
|
August 13, 2021
Discovery of ASTX029, A Clinical Candidate Which Modulates the Phosphorylation and Catalytic Activity of ERK1/2
Tom D Heightman, Valerio Berdini, Luke Bevan, et al.
Journal of Medicinal Chemistry
|
May 19, 2018
Fragment-Based Discovery of a Potent, Orally Bioavailable Inhibitor That Modulates the Phosphorylation and Catalytic Activity of ERK1/2
Tom D Heightman, Valerio Berdini, Hannah Braithwaite, et al.
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of 4
Search research articles
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Showing results (31-40 of 38) with videos related to
Sort By:
Page
of 4
You have reached the last page of results.
This site can display upto 38 results.
Molecular Cancer Therapeutics
|
August 14, 2021
Clinical Positioning of the IAP Antagonist Tolinapant (ASTX660) in Colorectal Cancer
Nyree Crawford, Katie J Stott, Tamas Sessler, et al.
Molecular Cancer Therapeutics
|
May 12, 2012
Chemosensitization of cancer cells by KU-0060648, a dual inhibitor of DNA-PK and PI-3K
Joanne M Munck, Michael A Batey, Yan Zhao, et al.
ACS Medicinal Chemistry Letters
|
July 21, 2015
Fragment-Based Discovery of Potent and Selective DDR1/2 Inhibitors
Christopher W Murray, Valerio Berdini, Ildiko M Buck, et al.
Journal of Medicinal Chemistry
|
August 10, 2018
A Fragment-Derived Clinical Candidate for Antagonism of X-Linked and Cellular Inhibitor of Apoptosis Proteins: 1-(6-[(4-Fluorophenyl)methyl]-5-(hydroxymethyl)-3,3-dimethyl-1 H,2 H,3 H-pyrrolo[3,2- b]pyridin-1-yl)-2-[(2 R,5 R)-5-methyl-2-([(3R)-3-methylmorpholin-4-yl]methyl)piperazin-1-yl]ethan-1-one (ASTX660)
Christopher N Johnson, Jong Sook Ahn, Ildiko M Buck, et al.
The Journal of Clinical Investigation
|
October 4, 2019
Selective DNA-PKcs inhibition extends the therapeutic index of localized radiotherapy and chemotherapy
Catherine E Willoughby, Yanyan Jiang, Huw D Thomas, et al.
Molecular Cancer Therapeutics
|
July 31, 2021
ASTX029, a Novel Dual-mechanism ERK Inhibitor, Modulates Both the Phosphorylation and Catalytic Activity of ERK
Joanne M Munck, Valerio Berdini, Luke Bevan, et al.
Journal of Medicinal Chemistry
|
August 13, 2021
Discovery of ASTX029, A Clinical Candidate Which Modulates the Phosphorylation and Catalytic Activity of ERK1/2
Tom D Heightman, Valerio Berdini, Luke Bevan, et al.
Journal of Medicinal Chemistry
|
May 19, 2018
Fragment-Based Discovery of a Potent, Orally Bioavailable Inhibitor That Modulates the Phosphorylation and Catalytic Activity of ERK1/2
Tom D Heightman, Valerio Berdini, Hannah Braithwaite, et al.
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of 4