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M Paola Costi

Showing results (1-10 of 19) with videos related to

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European Journal of Medicinal Chemistry|May 29, 2007
Synthesis of N-(5,7-diamino-3-phenyl-quinoxalin-2-yl)-3,4,5-substituted anilines and N-[4[(5,7-diamino-3-phenylquinoxalin-2-yl)amino]benzoyl]-l-glutamic acid diethyl ester: evaluation of in vitro anti-cancer and anti-folate activitiesPaola Corona, Mario Loriga, M Paola Costi, et al.
Journal of Medicinal Chemistry|February 18, 2005
Improving specificity vs bacterial thymidylate synthases through N-dansyl modulation of didansyltyrosineDonatella Tondi, Alberto Venturelli, Stefania Ferrari, et al.
Experimental Parasitology|December 5, 2012
Biochemical effects of riluzole on Leishmania parasitesDavide Guerrieri, Stefania Ferrari, M Paola Costi, et al.
Bioorganic & Medicinal Chemistry Letters|January 1, 2013
Ligand-based discovery of N-(1,3-dioxo-1H,3H-benzo[de]isochromen-5-yl)-carboxamide and sulfonamide derivatives as thymidylate synthase A inhibitorsStefania Ferrari, Marco Ingrami, Fabrizia Soragni, et al.
Journal of the American Chemical Society|March 31, 2005
Structure-based optimization of a non-beta-lactam lead results in inhibitors that do not up-regulate beta-lactamase expression in cell cultureDonatella Tondi, Federica Morandi, Richard Bonnet, et al.
Protein Science : a Publication of the Protein Society|March 23, 2010
Dimer-monomer equilibrium of human thymidylate synthase monitored by fluorescence resonance energy transferFilippo Genovese, Stefania Ferrari, Giambattista Guaitoli, et al.
Bioorganic & Medicinal Chemistry Letters|July 1, 2004
Aza-boronic acids as non-beta-lactam inhibitors of AmpC-beta-lactamaseValentina Buzzoni, Jesus Blazquez, Stefania Ferrari, et al.
Journal of Medicinal Chemistry|June 24, 2011
Identification of the binding modes of N-phenylphthalimides inhibiting bacterial thymidylate synthase through X-ray crystallography screeningStefano Mangani, Laura Cancian, Rosalida Leone, et al.
Biochimica Et Biophysica Acta|June 27, 2002
Structure-based studies on species-specific inhibition of thymidylate synthaseM Paola Costi, Donatella Tondi, Marcella Rinaldi, et al.
Acta Crystallographica. Section D, Biological Crystallography|October 6, 2005
The structure of Cryptococcus neoformans thymidylate synthase suggests strategies for using target dynamics for species-specific inhibitionJanet S Finer-Moore, Amy C Anderson, Robert H O'Neil, et al.
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Showing results (1-10 of 19) with videos related to

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Pageof 2
European Journal of Medicinal Chemistry|May 29, 2007
Synthesis of N-(5,7-diamino-3-phenyl-quinoxalin-2-yl)-3,4,5-substituted anilines and N-[4[(5,7-diamino-3-phenylquinoxalin-2-yl)amino]benzoyl]-l-glutamic acid diethyl ester: evaluation of in vitro anti-cancer and anti-folate activitiesPaola Corona, Mario Loriga, M Paola Costi, et al.
Journal of Medicinal Chemistry|February 18, 2005
Improving specificity vs bacterial thymidylate synthases through N-dansyl modulation of didansyltyrosineDonatella Tondi, Alberto Venturelli, Stefania Ferrari, et al.
Experimental Parasitology|December 5, 2012
Biochemical effects of riluzole on Leishmania parasitesDavide Guerrieri, Stefania Ferrari, M Paola Costi, et al.
Bioorganic & Medicinal Chemistry Letters|January 1, 2013
Ligand-based discovery of N-(1,3-dioxo-1H,3H-benzo[de]isochromen-5-yl)-carboxamide and sulfonamide derivatives as thymidylate synthase A inhibitorsStefania Ferrari, Marco Ingrami, Fabrizia Soragni, et al.
Journal of the American Chemical Society|March 31, 2005
Structure-based optimization of a non-beta-lactam lead results in inhibitors that do not up-regulate beta-lactamase expression in cell cultureDonatella Tondi, Federica Morandi, Richard Bonnet, et al.
Protein Science : a Publication of the Protein Society|March 23, 2010
Dimer-monomer equilibrium of human thymidylate synthase monitored by fluorescence resonance energy transferFilippo Genovese, Stefania Ferrari, Giambattista Guaitoli, et al.
Bioorganic & Medicinal Chemistry Letters|July 1, 2004
Aza-boronic acids as non-beta-lactam inhibitors of AmpC-beta-lactamaseValentina Buzzoni, Jesus Blazquez, Stefania Ferrari, et al.
Journal of Medicinal Chemistry|June 24, 2011
Identification of the binding modes of N-phenylphthalimides inhibiting bacterial thymidylate synthase through X-ray crystallography screeningStefano Mangani, Laura Cancian, Rosalida Leone, et al.
Biochimica Et Biophysica Acta|June 27, 2002
Structure-based studies on species-specific inhibition of thymidylate synthaseM Paola Costi, Donatella Tondi, Marcella Rinaldi, et al.
Acta Crystallographica. Section D, Biological Crystallography|October 6, 2005
The structure of Cryptococcus neoformans thymidylate synthase suggests strategies for using target dynamics for species-specific inhibitionJanet S Finer-Moore, Amy C Anderson, Robert H O'Neil, et al.
Pageof 2