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Journal of Medicinal Chemistry|April 23, 2014
Discovery of daclatasvir, a pan-genotypic hepatitis C virus NS5A replication complex inhibitor with potent clinical effectMakonen Belema, Nicholas A MeanwellAntimicrobial Agents and Chemotherapy|December 30, 2015
Synergistic Activity of Combined NS5A InhibitorsDonald R O'Boyle, Peter T Nower, Min Gao, et al.Current Drug Targets. Infectious Disorders|March 16, 2006
Developments in antiviral drug design, discovery and development in 2004Nicholas A Meanwell, Makonen Belema, David J Carini, et al.Journal of Medicinal Chemistry|March 14, 2014
Discovery and development of hepatitis C virus NS5A replication complex inhibitorsMakonen Belema, Omar D Lopez, John A Bender, et al.Bioorganic & Medicinal Chemistry Letters|January 2, 2007
Synthesis and biological evaluation of 4-amino derivatives of benzimidazoquinoxaline, benzimidazoquinoline, and benzopyrazoloquinazoline as potent IKK inhibitorsFrancis Beaulieu, Carl Ouellet, Edward H Ruediger, et al.The Journal of General Virology|July 29, 2011
The effects of NS5A inhibitors on NS5A phosphorylation, polyprotein processing and localizationDike Qiu, Julie A Lemm, Donald R O'Boyle, et al.Bioorganic & Medicinal Chemistry Letters|June 2, 2007
Synthesis and structure-activity relationship of imidazo(1,2-a)thieno(3,2-e)pyrazines as IKK-beta inhibitorsMakonen Belema, Amy Bunker, Van N Nguyen, et al.Virology|July 31, 2013
Characterizations of HCV NS5A replication complex inhibitorsDonald R O'Boyle Ii, Jin-Hua Sun, Peter T Nower, et al.Bioorganic & Medicinal Chemistry Letters|June 28, 2013
HCV NS5A replication complex inhibitors. Part 5: discovery of potent and pan-genotypic glycinamide cap derivativesMakonen Belema, Van N Nguyen, Denis R St Laurent, et al.Drug Metabolism and Disposition: the Biological Fate of Chemicals|April 1, 2016
Biotransformation of Daclatasvir In Vitro and in Nonclinical Species: Formation of the Main Metabolite by Pyrrolidine δ-Oxidation and RearrangementWenying Li, Weiping Zhao, Xiaohong Liu, et al.Pageof 3