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Malkeet Kumar

Showing results (1-10 of 11) with videos related to

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Bioorganic & Medicinal Chemistry Letters|June 5, 2014
Synthesis of new verapamil analogues and their evaluation in combination with rifampicin against Mycobacterium tuberculosis and molecular docking studies in the binding site of efflux protein Rv1258cKawaljit Singh, Malkeet Kumar, Elumalai Pavadai, et al.
ACS Infectious Diseases|February 21, 2023
Pyrido-Dibemequine Metabolites Exhibit Improved Druglike Features, Inhibit Hemozoin Formation in <i>Plasmodium falciparum</i>, and Synergize with Clinical AntimalarialsJohn Okombo, Malkeet Kumar, Devasha Redhi, et al.
Bioorganic & Medicinal Chemistry Letters|December 17, 2011
Synthesis, docking and in vitro antimalarial evaluation of bifunctional hybrids derived from β-lactams and 7-chloroquinoline using click chemistryPardeep Singh, Parvesh Singh, Malkeet Kumar, et al.
ACS Infectious Diseases|October 15, 2016
Design, Synthesis, and Evaluation of Novel Hybrid Efflux Pump Inhibitors for Use against Mycobacterium tuberculosisMalkeet Kumar, Kawaljit Singh, Krupa Naran, et al.
ACS Medicinal Chemistry Letters|August 20, 2021
Structure-Activity Relationship Studies Reveal New Astemizole Analogues Active against <i>Plasmodium falciparum</i> In VitroDickson Mambwe, Malkeet Kumar, Richard Ferger, et al.
Bioorganic & Medicinal Chemistry|January 27, 2018
Reversed isoniazids: Design, synthesis and evaluation against Mycobacterium tuberculosisMalkeet Kumar, Kawaljit Singh, Andile H Ngwane, et al.
Antimicrobial Agents and Chemotherapy|December 9, 2015
New Verapamil Analogs Inhibit Intracellular Mycobacteria without Affecting the Functions of Mycobacterium-Specific T CellsGetahun Abate, Peter G Ruminiski, Malkeet Kumar, et al.
ACS Infectious Diseases|December 15, 2020
New Amidated 3,6-Diphenylated Imidazopyridazines with Potent Antiplasmodium Activity Are Dual Inhibitors of <i>Plasmodium</i> Phosphatidylinositol-4-kinase and cGMP-Dependent Protein KinasePeter Mubanga Cheuka, Luyanda Centani, Lauren B Arendse, et al.
Journal of Medicinal Chemistry|December 12, 2022
Novel 3-Trifluoromethyl-1,2,4-oxadiazole Analogues of Astemizole with Multi-stage Antiplasmodium Activity and <i>In Vivo</i> Efficacy in a <i>Plasmodium berghei</i> Mouse Malaria Infection ModelDickson Mambwe, Constance M Korkor, Amanda Mabhula, et al.
ACS Infectious Diseases|December 12, 2018
Multistage Antiplasmodium Activity of Astemizole Analogues and Inhibition of Hemozoin Formation as a Contributor to Their Mode of ActionMalkeet Kumar, John Okombo, Dickson Mambwe, et al.
Pageof 2

Showing results (1-10 of 11) with videos related to

Sort By:
Pageof 2
Bioorganic & Medicinal Chemistry Letters|June 5, 2014
Synthesis of new verapamil analogues and their evaluation in combination with rifampicin against Mycobacterium tuberculosis and molecular docking studies in the binding site of efflux protein Rv1258cKawaljit Singh, Malkeet Kumar, Elumalai Pavadai, et al.
ACS Infectious Diseases|February 21, 2023
Pyrido-Dibemequine Metabolites Exhibit Improved Druglike Features, Inhibit Hemozoin Formation in <i>Plasmodium falciparum</i>, and Synergize with Clinical AntimalarialsJohn Okombo, Malkeet Kumar, Devasha Redhi, et al.
Bioorganic & Medicinal Chemistry Letters|December 17, 2011
Synthesis, docking and in vitro antimalarial evaluation of bifunctional hybrids derived from β-lactams and 7-chloroquinoline using click chemistryPardeep Singh, Parvesh Singh, Malkeet Kumar, et al.
ACS Infectious Diseases|October 15, 2016
Design, Synthesis, and Evaluation of Novel Hybrid Efflux Pump Inhibitors for Use against Mycobacterium tuberculosisMalkeet Kumar, Kawaljit Singh, Krupa Naran, et al.
ACS Medicinal Chemistry Letters|August 20, 2021
Structure-Activity Relationship Studies Reveal New Astemizole Analogues Active against <i>Plasmodium falciparum</i> In VitroDickson Mambwe, Malkeet Kumar, Richard Ferger, et al.
Bioorganic & Medicinal Chemistry|January 27, 2018
Reversed isoniazids: Design, synthesis and evaluation against Mycobacterium tuberculosisMalkeet Kumar, Kawaljit Singh, Andile H Ngwane, et al.
Antimicrobial Agents and Chemotherapy|December 9, 2015
New Verapamil Analogs Inhibit Intracellular Mycobacteria without Affecting the Functions of Mycobacterium-Specific T CellsGetahun Abate, Peter G Ruminiski, Malkeet Kumar, et al.
ACS Infectious Diseases|December 15, 2020
New Amidated 3,6-Diphenylated Imidazopyridazines with Potent Antiplasmodium Activity Are Dual Inhibitors of <i>Plasmodium</i> Phosphatidylinositol-4-kinase and cGMP-Dependent Protein KinasePeter Mubanga Cheuka, Luyanda Centani, Lauren B Arendse, et al.
Journal of Medicinal Chemistry|December 12, 2022
Novel 3-Trifluoromethyl-1,2,4-oxadiazole Analogues of Astemizole with Multi-stage Antiplasmodium Activity and <i>In Vivo</i> Efficacy in a <i>Plasmodium berghei</i> Mouse Malaria Infection ModelDickson Mambwe, Constance M Korkor, Amanda Mabhula, et al.
ACS Infectious Diseases|December 12, 2018
Multistage Antiplasmodium Activity of Astemizole Analogues and Inhibition of Hemozoin Formation as a Contributor to Their Mode of ActionMalkeet Kumar, John Okombo, Dickson Mambwe, et al.
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