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Chemmedchem|September 27, 2006
Mapping the fluorophilicity of a hydrophobic pocket: synthesis and biological evaluation of tricyclic thrombin inhibitors directing fluorinated alkyl groups into the p pocketAnja Hoffmann-Röder, Eliane Schweizer, Jonas Egger, et al.Chemmedchem|August 4, 2020
The Critical Role of Passive Permeability in Designing Successful DrugsLi Di, Per Artursson, Alex Avdeef, et al.Chemistry (Weinheim an Der Bergstrasse, Germany)|June 28, 2012
From lin-benzoguanines to lin-benzohypoxanthines as ligands for Zymomonas mobilis tRNA-guanine transglycosylase: replacement of protein-ligand hydrogen bonding by importing water clustersLuzi Jakob Barandun, Florian Immekus, Philipp C Kohler, et al.Chemmedchem|August 8, 2006
A fluorine scan at the catalytic center of thrombin: C--F, C--OH, and C--OMe bioisosterism and fluorine effects on pKa and log D valuesEliane Schweizer, Anja Hoffmann-Röder, Kaspar Schärer, et al.Drug Discovery Today|January 25, 2012
Can we discover pharmacological promiscuity early in the drug discovery process?Jens-Uwe Peters, Jérôme Hert, Caterina Bissantz, et al.Langmuir : the ACS Journal of Surfaces and Colloids|January 11, 2007
Self-assembly, DNA complexation, and pH response of amphiphilic dendrimers for gene transfectionMarine Guillot-Nieckowski, Derk Joester, Meike Stöhr, et al.Journal of Medicinal Chemistry|September 19, 2017
Lactam-Stapled Cell-Penetrating Peptides: Cell Uptake and Membrane Binding PropertiesMarco J Klein, Samuel Schmidt, Parvesh Wadhwani, et al.Nature Reviews. Drug Discovery|July 31, 2010
Coexistence of passive and carrier-mediated processes in drug transportKiyohiko Sugano, Manfred Kansy, Per Artursson, et al.Drug Discovery Today|April 18, 2012
Evidence-based approach to assess passive diffusion and carrier-mediated drug transportLi Di, Per Artursson, Alex Avdeef, et al.Bioorganic & Medicinal Chemistry Letters|June 5, 2004
An aminomethylpyrimidine DPP-IV inhibitor with improved propertiesJens-Uwe Peters, Daniel Hunziker, Holger Fischer, et al.Pageof 5