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Marcin Drop

Showing results (1-10 of 9) with videos related to

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Biomolecules|February 25, 2023
The Constitutive Activity of Spinal 5-HT<sub>6</sub> Receptors Contributes to Diabetic Neuropathic Pain in RatsNazarine Mokhtar, Marcin Drop, Florian Jacquot, et al.
Bioorganic & Medicinal Chemistry|August 7, 2019
Novel multitarget 5-arylidenehydantoins with arylpiperazinealkyl fragment: Pharmacological evaluation and investigation of cytotoxicity and metabolic stabilityAnna Czopek, Adam Bucki, Marcin Kołaczkowski, et al.
Journal of Neurochemistry|August 4, 2025
5-HT<sub>6</sub> Receptor Inverse Agonists Modulate Diabetic Neuropathic Pain in Female Rats: Evidence for 5-HT<sub>6</sub> Receptor Constitutive ActivityNazarine Mokhtar, Marcin Drop, Lauriane Delay, et al.
Progress in Neurobiology|June 9, 2020
mTOR activation by constitutively active serotonin6 receptors as new paradigm in neuropathic pain and its treatmentPierre-Yves Martin, Stéphane Doly, Al Mahdy Hamieh, et al.
European Journal of Medicinal Chemistry|June 27, 2024
5-HT<sub>6</sub> receptor neutral antagonists protect astrocytes: A lesson from 2-phenylpyrrole derivativesMarcin Drop, Paulina Koczurkiewicz-Adamczyk, Ophélie Bento, et al.
ACS Chemical Neuroscience|March 22, 2019
Dual 5-HT<sub>6</sub> and D<sub>3</sub> Receptor Antagonists in a Group of 1<i>H</i>-Pyrrolo[3,2-<i>c</i>]quinolines with Neuroprotective and Procognitive ActivityKatarzyna Grychowska, Severine Chaumont-Dubel, Rafał Kurczab, et al.
European Journal of Medicinal Chemistry|September 19, 2020
A dual-acting 5-HT<sub>6</sub> receptor inverse agonist/MAO-B inhibitor displays glioprotective and pro-cognitive propertiesVittorio Canale, Katarzyna Grychowska, Rafał Kurczab, et al.
ACS Chemical Neuroscience|March 11, 2021
2-Phenyl-1<i>H</i>-pyrrole-3-carboxamide as a New Scaffold for Developing 5-HT<sub>6</sub> Receptor Inverse Agonists with Cognition-Enhancing ActivityMarcin Drop, Vittorio Canale, Séverine Chaumont-Dubel, et al.
Bioorganic Chemistry|August 8, 2021
Neuropathic pain-alleviating activity of novel 5-HT<sub>6</sub> receptor inverse agonists derived from 2-aryl-1H-pyrrole-3-carboxamideMarcin Drop, Florian Jacquot, Vittorio Canale, et al.
Pageof 1

Showing results (1-10 of 9) with videos related to

Sort By:
Pageof 1
Biomolecules|February 25, 2023
The Constitutive Activity of Spinal 5-HT<sub>6</sub> Receptors Contributes to Diabetic Neuropathic Pain in RatsNazarine Mokhtar, Marcin Drop, Florian Jacquot, et al.
Bioorganic & Medicinal Chemistry|August 7, 2019
Novel multitarget 5-arylidenehydantoins with arylpiperazinealkyl fragment: Pharmacological evaluation and investigation of cytotoxicity and metabolic stabilityAnna Czopek, Adam Bucki, Marcin Kołaczkowski, et al.
Journal of Neurochemistry|August 4, 2025
5-HT<sub>6</sub> Receptor Inverse Agonists Modulate Diabetic Neuropathic Pain in Female Rats: Evidence for 5-HT<sub>6</sub> Receptor Constitutive ActivityNazarine Mokhtar, Marcin Drop, Lauriane Delay, et al.
Progress in Neurobiology|June 9, 2020
mTOR activation by constitutively active serotonin6 receptors as new paradigm in neuropathic pain and its treatmentPierre-Yves Martin, Stéphane Doly, Al Mahdy Hamieh, et al.
European Journal of Medicinal Chemistry|June 27, 2024
5-HT<sub>6</sub> receptor neutral antagonists protect astrocytes: A lesson from 2-phenylpyrrole derivativesMarcin Drop, Paulina Koczurkiewicz-Adamczyk, Ophélie Bento, et al.
ACS Chemical Neuroscience|March 22, 2019
Dual 5-HT<sub>6</sub> and D<sub>3</sub> Receptor Antagonists in a Group of 1<i>H</i>-Pyrrolo[3,2-<i>c</i>]quinolines with Neuroprotective and Procognitive ActivityKatarzyna Grychowska, Severine Chaumont-Dubel, Rafał Kurczab, et al.
European Journal of Medicinal Chemistry|September 19, 2020
A dual-acting 5-HT<sub>6</sub> receptor inverse agonist/MAO-B inhibitor displays glioprotective and pro-cognitive propertiesVittorio Canale, Katarzyna Grychowska, Rafał Kurczab, et al.
ACS Chemical Neuroscience|March 11, 2021
2-Phenyl-1<i>H</i>-pyrrole-3-carboxamide as a New Scaffold for Developing 5-HT<sub>6</sub> Receptor Inverse Agonists with Cognition-Enhancing ActivityMarcin Drop, Vittorio Canale, Séverine Chaumont-Dubel, et al.
Bioorganic Chemistry|August 8, 2021
Neuropathic pain-alleviating activity of novel 5-HT<sub>6</sub> receptor inverse agonists derived from 2-aryl-1H-pyrrole-3-carboxamideMarcin Drop, Florian Jacquot, Vittorio Canale, et al.
Pageof 1