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Molecular Pharmaceutics|April 10, 2026
Nanostructured Lipid Carriers Enhance Brain Delivery and Antioxidant Efficacy of a Small-Molecule MAO B Inhibitor for Neurodegenerative Disease TherapyRita Mastrogiacomo, Daniela Valeria Miniero, Mariagrazia Rullo, et al.ACS Medicinal Chemistry Letters|May 22, 2020
Chiral Separation, X-ray Structure, and Biological Evaluation of a Potent and Reversible Dual Binding Site AChE InhibitorMarco Catto, Leonardo Pisani, Eugenio de la Mora, et al.Journal of Medicinal Chemistry|June 25, 2015
Structure-Based Design and Optimization of Multitarget-Directed 2H-Chromen-2-one Derivatives as Potent Inhibitors of Monoamine Oxidase B and CholinesterasesRoberta Farina, Leonardo Pisani, Marco Catto, et al.European Journal of Medicinal Chemistry|February 8, 2023
Thioxanthenone-based derivatives as multitarget therapeutic leads for Alzheimer's diseaseMichele Tonelli, Marco Catto, Raimon Sabaté, et al.European Journal of Pharmaceutical Sciences : Official Journal of the European Federation for Pharmaceutical Sciences|March 10, 2025
Light-mediated activation/deactivation control and in vitro ADME-Tox profiling of a donepezil-like Dual AChE/MAO-B InhibitorFederica Poggialini, Paolo Governa, Chiara Vagaggini, et al.Archiv Der Pharmazie|December 29, 2023
Radiosynthesis and whole-body distribution in mice of a <sup>18</sup> F-labeled azepino[4,3-b]indole-1-one derivative with multimodal activity for the treatment of Alzheimer's diseaseSang Hee Lee, Rosa Purgatorio, Francesco Samarelli, et al.European Journal of Medicinal Chemistry|March 15, 2024
Novel 6-hydroxybenzothiazol-2-carboxamides as potent and selective monoamine oxidase B inhibitors endowed with neuroprotective activityOmar M Al-Saad, Moustafa Gabr, Sarah S Darwish, et al.Pharmaceuticals (Basel, Switzerland)|April 27, 2024
Nature-Inspired 1-Phenylpyrrolo[2,1-<i>a</i>]isoquinoline Scaffold for Novel Antiproliferative Agents Circumventing P-Glycoprotein-Dependent Multidrug ResistanceAlisa A Nevskaya, Rosa Purgatorio, Tatiana N Borisova, et al.Molecules (Basel, Switzerland)|January 15, 2021
Homobivalent Lamellarin-Like Schiff Bases: In Vitro Evaluation of Their Cancer Cell Cytotoxicity and Multitargeting Anti-Alzheimer's Disease PotentialAlisa A Nevskaya, Lada V Anikina, Rosa Purgatorio, et al.RSC Medicinal Chemistry|December 10, 2025
Exploring pyrazolidinone and pyrazolidinedione scaffolds for Alzheimer's therapy: multitarget COX-2 inhibitors with anti-amyloid β, anti-tau, antioxidant, and neuroprotective activitiesMichael Emad, Reham Waheed, Zeinab Mostafa, et al.Pageof 12