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Nature Reviews. Drug Discovery|July 18, 2002
The potential for novel anti-inflammatory therapies for coronary artery diseaseMargaret A Cascieri
Bioorganic & Medicinal Chemistry Letters|May 8, 2007
3-Amino-1-alkyl-cyclopentane carboxamides as small molecule antagonists of the human and murine CC chemokine receptor 2Gabor Butora, Richard Jiao, William H Parsons, et al.
Gene|October 18, 2002
Identification, localization and receptor characterization of novel mammalian substance P-like peptidesMarc M Kurtz, Ruiping Wang, Michelle K Clements, et al.
Bioorganic & Medicinal Chemistry Letters|July 28, 2006
4-Amino-2-alkyl-butyramides as small molecule CCR2 antagonists with favorable pharmacokinetic propertiesGabor Butora, Gregori J Morriello, Shankaran Kothandaraman, et al.
Bioorganic & Medicinal Chemistry Letters|November 10, 2006
Alpha-aminothiazole-gamma-aminobutanoic amides as potent, small molecule CCR2 receptor antagonistsChangyou Zhou, Liangqin Guo, William H Parsons, et al.
Biochemical Pharmacology|June 27, 2003
Expression and characterization of the chemokine receptor CCR2B from rhesus monkeyHong Jin, Pasquale P Vicario, Hans Zweerink, et al.
Journal of Medicinal Chemistry|April 28, 2007
Discovery of 3-piperidinyl-1-cyclopentanecarboxamide as a novel scaffold for highly potent CC chemokine receptor 2 antagonistsLihu Yang, Gabor Butora, Richard X Jiao, et al.
Bioorganic & Medicinal Chemistry Letters|September 10, 2002
Spirocyclic NK(1) antagonists II: [4.5]-spiroethersBrian J Williams, Margaret A Cascieri, Gary G Chicchi, et al.
Bioorganic & Medicinal Chemistry Letters|July 11, 2006
Cyclopentane-based human NK1 antagonists. Part 1: discovery and initial SARPaul E Finke, Laura C Meurer, Dorothy A Levorse, et al.
Bioorganic & Medicinal Chemistry Letters|May 16, 2006
Discovery of 3,5-bis(trifluoromethyl)benzyl L-arylglycinamide based potent CCR2 antagonistsLihu Yang, Changyou Zhou, Liangqin Guo, et al.
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