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Frontiers in Cellular and Infection Microbiology|June 27, 2022
Adapt or Die: Targeting Unique Transmission-Stage Biology for Malaria EliminationMariëtte E van der Watt, Janette Reader, Lyn-Marié BirkholtzJournal of Ethnopharmacology|July 19, 2022
In vitro dual activity of Aloe marlothii roots and its chemical constituents against Plasmodium falciparum asexual and sexual stage parasitesSephora Mutombo Mianda, Luke Invernizzi, Mariëtte E van der Watt, et al.Pharmaceutics|December 28, 2021
The Artemiside-Artemisox-Artemisone-M1 Tetrad: Efficacies against Blood Stage P. falciparum Parasites, DMPK Properties, and the Case for ArtemisideLiezl Gibhard, Dina Coertzen, Janette Reader, et al.International Journal for Parasitology. Drugs and Drug Resistance|June 7, 2020
Naphthylisoquinoline alkaloids, validated as hit multistage antiplasmodial natural productsPhanankosi Moyo, William Shamburger, Mariëtte E van der Watt, et al.Chembiochem : a European Journal of Chemical Biology|September 15, 2022
New Transmission-Selective Antimalarial Agents through Hit-to-Lead Optimization of 2-([1,1'-Biphenyl]-4-carboxamido)benzoic Acid DerivativesJanette Reader, Daniel F L Opperman, Mariëtte E van der Watt, et al.Frontiers in Chemistry|January 31, 2020
Optimal 10-Aminoartemisinins With Potent Transmission-Blocking Capabilities for New Artemisinin Combination Therapies-Activities Against Blood Stage P. falciparum Including PfKI3 C580Y Mutants and Liver Stage P. berghei ParasitesHo Ning Wong, Vivian Padín-Irizarry, Mariëtte E van der Watt, et al.ACS Infectious Diseases|August 14, 2024
The Tuberculosis Drug Candidate SQ109 and Its Analogs Have Multistage Activity against Plasmodium falciparumSavannah J Watson, Mariëtte E van der Watt, Anjo Theron, et al.The Journal of Antimicrobial Chemotherapy|February 9, 2018
Potent Plasmodium falciparum gametocytocidal compounds identified by exploring the kinase inhibitor chemical space for dual active antimalarialsMariëtte E van der Watt, Janette Reader, Alisje Churchyard, et al.Nature Communications|January 12, 2021
Multistage and transmission-blocking targeted antimalarials discovered from the open-source MMV Pandemic Response BoxJanette Reader, Mariëtte E van der Watt, Dale Taylor, et al.Antimicrobial Agents and Chemotherapy|June 27, 2018
UCT943, a Next-Generation Plasmodium falciparum PI4K Inhibitor Preclinical Candidate for the Treatment of MalariaChristel Brunschwig, Nina Lawrence, Dale Taylor, et al.Pageof 1