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European Journal of Medicinal Chemistry|October 15, 2017
Crassiflorone derivatives that inhibit Trypanosoma brucei glyceraldehyde-3-phosphate dehydrogenase (TbGAPDH) and Trypanosoma cruzi trypanothione reductase (TcTR) and display trypanocidal activityElisa Uliassi, Giulia Fiorani, R Luise Krauth-Siegel, et al.Chemmedchem|December 25, 2014
Novel tacrine-grafted Ugi adducts as multipotent anti-Alzheimer drugs: a synthetic renewal in tacrine-ferulic acid hybridsMohamed Benchekroun, Manuela Bartolini, Javier Egea, et al.ACS Chemical Neuroscience|July 22, 2022
Riluzole-Rasagiline Hybrids: Toward the Development of Multi-Target-Directed Ligands for Amyotrophic Lateral SclerosisClaudia Albertini, Alessandra Salerno, Silvia Atzeni, et al.European Journal of Medicinal Chemistry|August 21, 2021
From virtual screening hits targeting a cryptic pocket in BACE-1 to a nontoxic brain permeable multitarget anti-Alzheimer lead with disease-modifying and cognition-enhancing effectsCaterina Pont, Tiziana Ginex, Christian Griñán-Ferré, et al.European Journal of Medicinal Chemistry|January 27, 2020
Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaignPasquale Linciano, Gregorio Cullia, Chiara Borsari, et al.European Journal of Medicinal Chemistry|January 7, 2016
Cardanol-derived AChE inhibitors: Towards the development of dual binding derivatives for Alzheimer's diseaseLaís Flávia Nunes Lemes, Giselle de Andrade Ramos, Andressa Souza de Oliveira, et al.ACS Medicinal Chemistry Letters|April 17, 2024
Empowering Voices: Inspiring Women in Medicinal ChemistryMaria-Jesus Blanco, Joanne J Bronson, Erin F DiMauro, et al.Journal of Medicinal Chemistry|March 8, 2024
Empowering Voices: Inspiring Women in Medicinal ChemistryMaria-Jesus Blanco, Joanne J Bronson, Erin F DiMauro, et al.European Journal of Medicinal Chemistry|March 10, 2019
Novel tacrine-tryptophan hybrids: Multi-target directed ligands as potential treatment for Alzheimer's diseaseKatarina Chalupova, Jan Korabecny, Manuela Bartolini, et al.ACS Medicinal Chemistry Letters|September 18, 2024
Benign-by-Design SAHA Analogues for Human and Animal Vector-Borne Parasitic DiseasesMichele Rossi, Bianca Martinengo, Eleonora Diamanti, et al.Pageof 14