Showing results (81-90 of 113) with videos related to
Sort By:
Pageof 12
Computers in Biology and Medicine|April 23, 2024
DeLA-DrugSelf: Empowering multi-objective de novo design through SELFIES molecular representationDomenico Alberga, Giuseppe Lamanna, Giovanni Graziano, et al.Bioorganic & Medicinal Chemistry|October 16, 2007
Small P-gp modulating molecules: SAR studies on tetrahydroisoquinoline derivativesNicola Antonio Colabufo, Francesco Berardi, Mariangela Cantore, et al.Journal of Medicinal Chemistry|December 26, 2018
Design, Biological Evaluation, and Molecular Modeling of Tetrahydroisoquinoline Derivatives: Discovery of A Potent P-Glycoprotein Ligand Overcoming Multidrug Resistance in Cancer Stem CellsChiara Riganti, Marialessandra Contino, Stefano Guglielmo, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|April 8, 2020
6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline amides and corresponding ester isosteres as multidrug resistance reversersLaura Braconi, Gianluca Bartolucci, Marialessandra Contino, et al.Molecules (Basel, Switzerland)|July 27, 2024
Dual Inhibitors of P-gp and Carbonic Anhydrase XII (hCA XII) against Tumor Multidrug Resistance with Piperazine ScaffoldLaura Braconi, Chiara Riganti, Astrid Parenti, et al.Medchemcomm|August 16, 2018
New tetrahydroisoquinoline-based P-glycoprotein modulators: decoration of the biphenyl core gives selective ligandsMarialessandra Contino, Stefano Guglielmo, Maria Grazia Perrone, et al.Journal of Medicinal Chemistry|March 15, 2023
Development of Fluorescent 4-[4-(3H-Spiro[isobenzofuran-1,4'-piperidin]-1'-yl)butyl]indolyl Derivatives as High-Affinity Probes to Enable the Study of σ Receptors via Fluorescence-Based TechniquesFrancesca Serena Abatematteo, Maria Majellaro, Bianca Montsch, et al.European Journal of Medicinal Chemistry|October 15, 2023
Development of potent isoflavone-based formyl peptide receptor 1 (FPR1) antagonists and their effects in gastric cancer cell modelsFabio Francavilla, Federica Sarcina, Igor A Schepetkin, et al.Journal of Medicinal Chemistry|April 12, 2011
Novel potent and selective σ ligands: evaluation of their agonist and antagonist propertiesAgostino Marrazzo, Enrique J Cobos, Carmela Parenti, et al.International Journal of Pharmaceutics|October 29, 2020
Induced expression of P-gp and BCRP transporters on brain endothelial cells using transferrin functionalized nanostructured lipid carriers: A first step of a potential strategy for the treatment of Alzheimer's diseaseIlaria Arduino, Rosa Maria Iacobazzi, Chiara Riganti, et al.Pageof 12