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Bioorganic & Medicinal Chemistry Letters
|
May 20, 2011
Indole 5-carboxamide Thumb Pocket I inhibitors of HCV NS5B polymerase with nanomolar potency in cell-based subgenomic replicons (part 2): central amino acid linker and right-hand-side SAR studies
Pierre L Beaulieu, Catherine Chabot, Jianmin Duan, et al.
Angewandte Chemie (International Ed. in English)
|
September 16, 2004
Binding mode determination of benzimidazole inhibitors of the hepatitis C virus RNA polymerase by a structure and dynamics strategy
Steven R LaPlante, Araz Jakalian, Norman Aubry, et al.
Journal of Medicinal Chemistry
|
October 29, 2013
Conformation-based restrictions and scaffold replacements in the design of hepatitis C virus polymerase inhibitors: discovery of deleobuvir (BI 207127)
Steven R LaPlante, Michael Bös, Christian Brochu, et al.
Journal of Medicinal Chemistry
|
August 2, 2012
Discovery of the first thumb pocket 1 NS5B polymerase inhibitor (BILB 1941) with demonstrated antiviral activity in patients chronically infected with genotype 1 hepatitis C virus (HCV)
Pierre L Beaulieu, Michael Bös, Michael G Cordingley, et al.
Bioorganic & Medicinal Chemistry Letters
|
June 18, 2013
Structure-based design of novel HCV NS5B thumb pocket 2 allosteric inhibitors with submicromolar gt1 replicon potency: discovery of a quinazolinone chemotype
Pierre L Beaulieu, René Coulombe, Jianmin Duan, et al.
Organic Letters
|
August 28, 2004
Synthesis of BILN 2061, an HCV NS3 protease inhibitor with proven antiviral effect in humans
Anne-Marie Faucher, Murray D Bailey, Pierre L Beaulieu, et al.
Plos One
|
April 8, 2022
Development of mAb-based polyglutamine-dependent and polyglutamine length-independent huntingtin quantification assays with cross-site validation
David F Fischer, Sipke Dijkstra, Kimberly Lo, et al.
Journal of Medicinal Chemistry
|
March 19, 2004
Structure-activity study on a novel series of macrocyclic inhibitors of the hepatitis C virus NS3 protease leading to the discovery of BILN 2061
Montse Llinàs-Brunet, Murray D Bailey, Gordon Bolger, et al.
Journal of Medicinal Chemistry
|
June 19, 2013
Molecular dynamics simulations and structure-based rational design lead to allosteric HCV NS5B polymerase thumb pocket 2 inhibitor with picomolar cellular replicon potency
Oliver Hucke, René Coulombe, Pierre Bonneau, et al.
Bioorganic & Medicinal Chemistry Letters
|
January 16, 2010
N-Acetamideindolecarboxylic acid allosteric 'finger-loop' inhibitors of the hepatitis C virus NS5B polymerase: discovery and initial optimization studies
Pierre L Beaulieu, Eric Jolicoeur, James Gillard, et al.
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Search research articles
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Showing results (11-20 of 22) with videos related to
Sort By:
Page
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Bioorganic & Medicinal Chemistry Letters
|
May 20, 2011
Indole 5-carboxamide Thumb Pocket I inhibitors of HCV NS5B polymerase with nanomolar potency in cell-based subgenomic replicons (part 2): central amino acid linker and right-hand-side SAR studies
Pierre L Beaulieu, Catherine Chabot, Jianmin Duan, et al.
Angewandte Chemie (International Ed. in English)
|
September 16, 2004
Binding mode determination of benzimidazole inhibitors of the hepatitis C virus RNA polymerase by a structure and dynamics strategy
Steven R LaPlante, Araz Jakalian, Norman Aubry, et al.
Journal of Medicinal Chemistry
|
October 29, 2013
Conformation-based restrictions and scaffold replacements in the design of hepatitis C virus polymerase inhibitors: discovery of deleobuvir (BI 207127)
Steven R LaPlante, Michael Bös, Christian Brochu, et al.
Journal of Medicinal Chemistry
|
August 2, 2012
Discovery of the first thumb pocket 1 NS5B polymerase inhibitor (BILB 1941) with demonstrated antiviral activity in patients chronically infected with genotype 1 hepatitis C virus (HCV)
Pierre L Beaulieu, Michael Bös, Michael G Cordingley, et al.
Bioorganic & Medicinal Chemistry Letters
|
June 18, 2013
Structure-based design of novel HCV NS5B thumb pocket 2 allosteric inhibitors with submicromolar gt1 replicon potency: discovery of a quinazolinone chemotype
Pierre L Beaulieu, René Coulombe, Jianmin Duan, et al.
Organic Letters
|
August 28, 2004
Synthesis of BILN 2061, an HCV NS3 protease inhibitor with proven antiviral effect in humans
Anne-Marie Faucher, Murray D Bailey, Pierre L Beaulieu, et al.
Plos One
|
April 8, 2022
Development of mAb-based polyglutamine-dependent and polyglutamine length-independent huntingtin quantification assays with cross-site validation
David F Fischer, Sipke Dijkstra, Kimberly Lo, et al.
Journal of Medicinal Chemistry
|
March 19, 2004
Structure-activity study on a novel series of macrocyclic inhibitors of the hepatitis C virus NS3 protease leading to the discovery of BILN 2061
Montse Llinàs-Brunet, Murray D Bailey, Gordon Bolger, et al.
Journal of Medicinal Chemistry
|
June 19, 2013
Molecular dynamics simulations and structure-based rational design lead to allosteric HCV NS5B polymerase thumb pocket 2 inhibitor with picomolar cellular replicon potency
Oliver Hucke, René Coulombe, Pierre Bonneau, et al.
Bioorganic & Medicinal Chemistry Letters
|
January 16, 2010
N-Acetamideindolecarboxylic acid allosteric 'finger-loop' inhibitors of the hepatitis C virus NS5B polymerase: discovery and initial optimization studies
Pierre L Beaulieu, Eric Jolicoeur, James Gillard, et al.
Page
of 3