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Journal of Medicinal Chemistry|September 26, 2018
Design, Synthesis, and Evaluation of Piperazinyl Pyrrolidin-2-ones as a Novel Series of Reversible Monoacylglycerol Lipase InhibitorsJumpei Aida, Makoto Fushimi, Tomokazu Kusumoto, et al.The Journal of Pharmacology and Experimental Therapeutics|September 18, 2021
Selective Acetyl-CoA Carboxylase 1 Inhibitor Improves Hepatic Steatosis and Hepatic Fibrosis in a Preclinical Nonalcoholic Steatohepatitis ModelYumiko Okano Tamura, Jun Sugama, Shinji Iwasaki, et al.Lab on a Chip|May 30, 2025
A polystyrene-film-based device for engineered cardiac tissues enables accurate analysis of drug responses on contractile propertiesYuya Fujiwara, Masako Sasaki, Sohei Funaoka, et al.Journal of Medicinal Chemistry|December 13, 2017
Discovery of Novel Selective Acetyl-CoA Carboxylase (ACC) 1 InhibitorsRyo Mizojiri, Moriteru Asano, Daisuke Tomita, et al.Stem Cell Reports|October 6, 2023
ERRγ agonist under mechanical stretching manifests hypertrophic cardiomyopathy phenotypes of engineered cardiac tissue through maturationYuya Fujiwara, Kenji Miki, Kohei Deguchi, et al.Scientific Reports|October 1, 2013
In situ label-free imaging for visualizing the biotransformation of a bioactive polyphenolYoon Hee Kim, Yoshinori Fujimura, Takatoki Hagihara, et al.Bioorganic & Medicinal Chemistry Letters|June 9, 2012
Symmetrical approach of spiro-pyrazolidinediones as acetyl-CoA carboxylase inhibitorsMakoto Kamata, Tohru Yamashita, Asato Kina, et al.Pharmacology Research & Perspectives|September 12, 2019
Discovery and characterization of a small-molecule enteropeptidase inhibitor, SCO-792Masako Sasaki, Ikuo Miyahisa, Sachiko Itono, et al.Journal of Medicinal Chemistry|February 13, 2019
Design, Synthesis, and Evaluation of (4 R)-1-{3-[2-(18F)Fluoro-4-methylpyridin-3-yl]phenyl}-4-[4-(1,3-thiazol-2-ylcarbonyl)piperazin-1-yl]pyrrolidin-2-one ([18F]T-401) as a Novel Positron-Emission Tomography Imaging Agent for Monoacylglycerol LipaseYasushi Hattori, Kazunobu Aoyama, Jun Maeda, et al.Scientific Reports|September 27, 2013
Green tea extract containing a highly absorbent catechin prevents diet-induced lipid metabolism disorderTakashi Suzuki, Motofumi Kumazoe, Yoonhee Kim, et al.Pageof 5