Jove
Visualize
Contact Us
JoVE
x logofacebook logolinkedin logoyoutube logo
ABOUT JoVE
OverviewLeadershipBlogJoVE Help Center
AUTHORS
Publishing ProcessEditorial BoardScope & PoliciesPeer ReviewFAQSubmit
LIBRARIANS
TestimonialsSubscriptionsAccessResourcesLibrary Advisory BoardFAQ
RESEARCH
JoVE JournalMethods CollectionsJoVE Encyclopedia of ExperimentsArchive
EDUCATION
JoVE CoreJoVE BusinessJoVE Science EducationJoVE Lab ManualFaculty Resource CenterFaculty Site
Terms & Conditions of Use
Privacy Policy
Policies

Filters

Matthias Engel

Showing results (41-50 of 79) with videos related to

Pageof 8
Sort By:
European Journal of Medicinal Chemistry|October 28, 2021
Discovery of novel 6-hydroxybenzothiazole urea derivatives as dual Dyrk1A/α-synuclein aggregation inhibitors with neuroprotective effectsYasmeen T AlNajjar, Moustafa Gabr, Ahmed K ElHady, et al.
Journal of Medicinal Chemistry|August 26, 2011
4-benzimidazolyl-3-phenylbutanoic acids as novel PIF-pocket-targeting allosteric inhibitors of protein kinase PKCζWolfgang Fröhner, Laura A Lopez-Garcia, Sonja Neimanis, et al.
Journal of Medicinal Chemistry|January 29, 2019
2-Aminothiazole Derivatives as Selective Allosteric Modulators of the Protein Kinase CK2. 2. Structure-Based Optimization and Investigation of Effects Specific to the Allosteric Mode of ActionBenoît Bestgen, Irina Kufareva, Weiguang Seetoh, et al.
ACS Chemical Biology|August 6, 2013
PIF-pocket as a target for C. albicans Pkh selective inhibitorsDaniel Pastor-Flores, Jörg O Schulze, Anna Bahí, et al.
Journal of Medicinal Chemistry|October 31, 2012
2-(3-Oxo-1,3-diphenylpropyl)malonic acids as potent allosteric ligands of the PIF pocket of phosphoinositide-dependent kinase-1: development and prodrug conceptAdriana Wilhelm, Laura A Lopez-Garcia, Katrien Busschots, et al.
Cancers|June 19, 2024
<i>N</i>-Benzylated 5-Hydroxybenzothiophene-2-carboxamides as Multi-Targeted Clk/Dyrk Inhibitors and Potential Anticancer AgentsNoha Mostafa, Po-Jen Chen, Sarah S Darwish, et al.
Pharmaceuticals (Basel, Switzerland)|July 27, 2022
Development of (4-Phenylamino)quinazoline Alkylthiourea Derivatives as Novel NF-κB InhibitorsSarah S Darwish, Po-Jen Chen, Mostafa M Hamed, et al.
The Journal of Biological Chemistry|September 3, 2009
Regulation of the interaction between protein kinase C-related protein kinase 2 (PRK2) and its upstream kinase, 3-phosphoinositide-dependent protein kinase 1 (PDK1)Rosalia Dettori, Silvina Sonzogni, Lucas Meyer, et al.
The Journal of Biological Chemistry|July 13, 2024
Molecular insights into the regulatory landscape of PKC-related kinase-2 (PRK2/PKN2) using targeted small compoundsLissy Z F Gross, Angelika F Winkel, Facundo Galceran, et al.
Bioorganic Chemistry|July 2, 2022
From EGFR kinase inhibitors to anti-inflammatory drugs: Optimization and biological evaluation of (4-(phenylamino)quinazolinyl)-phenylthiourea derivatives as novel NF-κB inhibitorsReem A Wagdy, Po-Jen Chen, Mostafa M Hamed, et al.
Pageof 8

Showing results (41-50 of 79) with videos related to

Sort By:
Pageof 8
European Journal of Medicinal Chemistry|October 28, 2021
Discovery of novel 6-hydroxybenzothiazole urea derivatives as dual Dyrk1A/α-synuclein aggregation inhibitors with neuroprotective effectsYasmeen T AlNajjar, Moustafa Gabr, Ahmed K ElHady, et al.
Journal of Medicinal Chemistry|August 26, 2011
4-benzimidazolyl-3-phenylbutanoic acids as novel PIF-pocket-targeting allosteric inhibitors of protein kinase PKCζWolfgang Fröhner, Laura A Lopez-Garcia, Sonja Neimanis, et al.
Journal of Medicinal Chemistry|January 29, 2019
2-Aminothiazole Derivatives as Selective Allosteric Modulators of the Protein Kinase CK2. 2. Structure-Based Optimization and Investigation of Effects Specific to the Allosteric Mode of ActionBenoît Bestgen, Irina Kufareva, Weiguang Seetoh, et al.
ACS Chemical Biology|August 6, 2013
PIF-pocket as a target for C. albicans Pkh selective inhibitorsDaniel Pastor-Flores, Jörg O Schulze, Anna Bahí, et al.
Journal of Medicinal Chemistry|October 31, 2012
2-(3-Oxo-1,3-diphenylpropyl)malonic acids as potent allosteric ligands of the PIF pocket of phosphoinositide-dependent kinase-1: development and prodrug conceptAdriana Wilhelm, Laura A Lopez-Garcia, Katrien Busschots, et al.
Cancers|June 19, 2024
<i>N</i>-Benzylated 5-Hydroxybenzothiophene-2-carboxamides as Multi-Targeted Clk/Dyrk Inhibitors and Potential Anticancer AgentsNoha Mostafa, Po-Jen Chen, Sarah S Darwish, et al.
Pharmaceuticals (Basel, Switzerland)|July 27, 2022
Development of (4-Phenylamino)quinazoline Alkylthiourea Derivatives as Novel NF-κB InhibitorsSarah S Darwish, Po-Jen Chen, Mostafa M Hamed, et al.
The Journal of Biological Chemistry|September 3, 2009
Regulation of the interaction between protein kinase C-related protein kinase 2 (PRK2) and its upstream kinase, 3-phosphoinositide-dependent protein kinase 1 (PDK1)Rosalia Dettori, Silvina Sonzogni, Lucas Meyer, et al.
The Journal of Biological Chemistry|July 13, 2024
Molecular insights into the regulatory landscape of PKC-related kinase-2 (PRK2/PKN2) using targeted small compoundsLissy Z F Gross, Angelika F Winkel, Facundo Galceran, et al.
Bioorganic Chemistry|July 2, 2022
From EGFR kinase inhibitors to anti-inflammatory drugs: Optimization and biological evaluation of (4-(phenylamino)quinazolinyl)-phenylthiourea derivatives as novel NF-κB inhibitorsReem A Wagdy, Po-Jen Chen, Mostafa M Hamed, et al.
Pageof 8