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Journal of Medicinal Chemistry|October 18, 2013
The versatile nature of the 6-aminoquinolone scaffold: identification of submicromolar hepatitis C virus NS5B inhibitorsGiuseppe Manfroni, Rolando Cannalire, Maria Letizia Barreca, et al.Cell Reports|August 2, 2018
Noelin1 Affects Lateral Mobility of Synaptic AMPA ReceptorsNikhil J Pandya, Christian Seeger, Norbert Babai, et al.Nucleic Acids Research|August 12, 2025
Deciphering the RNA recognition by Musashi-1 to design protein and RNA variants for in vitro and in vivo applicationsAnna Pérez-Ràfols, Guillermo Pérez-Ropero, Linda Cerofolini, et al.ACS Medicinal Chemistry Letters|February 18, 2026
Discovery of Potent, Selective, and Brain-Penetrant Small Molecule CD38 InhibitorsAndrew J Stott, Roland W Bürli, Kevin J Doyle, et al.Nucleic Acids Research|October 3, 2022
Monitoring drug-target interactions through target engagement-mediated amplification on arrays and in situRasel A Al-Amin, Lars Johansson, Eldar Abdurakhmanov, et al.SLAS Discovery : Advancing Life Sciences R & D|September 15, 2023
Multiplexed experimental strategies for fragment library screening against challenging drug targets using SPR biosensorsEdward A FitzGerald, Darius Vagrys, Giulia Opassi, et al.Nature Communications|June 13, 2015
Proximity-dependent initiation of hybridization chain reactionBjörn Koos, Gaëlle Cane, Karin Grannas, et al.Chemmedchem|August 28, 2024
The Role of Water Networks in Phosphodiesterase Inhibitor Dissociation and Kinetic SelectivityAntoni R Blaazer, Abhimanyu K Singh, Lorena Zara, et al.Chembiochem : a European Journal of Chemical Biology|January 5, 2021
Discovery of an Allosteric Ligand Binding Site in SMYD3 Lysine MethyltransferaseVladimir O Talibov, Edoardo Fabini, Edward A FitzGerald, et al.European Journal of Medicinal Chemistry|September 18, 2022
Discovery of the 4-aminopiperidine-based compound EM127 for the site-specific covalent inhibition of SMYD3Marco Daniele Parenti, Marina Naldi, Elisabetta Manoni, et al.Pageof 13