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Journal of Medicinal Chemistry|October 27, 2006
Further studies on imidazo[4,5-b]pyridine AT1 angiotensin II receptor antagonists. Effects of the transformation of the 4-phenylquinoline backbone into 4-phenylisoquinolinone or 1-phenylindene scaffoldsAndrea Cappelli, Gal la Pericot Mohr, Germano Giuliani, et al.Bioorganic & Medicinal Chemistry|January 19, 2015
Synthesis, biological evaluation and docking analysis of a new series of methylsulfonyl and sulfamoyl acetamides and ethyl acetates as potent COX-2 inhibitorsSara Consalvi, Salvatore Alfonso, Angela Di Capua, et al.Journal of Medicinal Chemistry|April 30, 2004
Design, synthesis, structural studies, biological evaluation, and computational simulations of novel potent AT(1) angiotensin II receptor antagonists based on the 4-phenylquinoline structureAndrea Cappelli, Gal la Pericot Mohr Gl, Andrea Gallelli, et al.European Journal of Medicinal Chemistry|December 7, 2016
Synthesis and biological evaluation of a new class of benzothiazines as neuroprotective agentsAlessandra Mancini, Alessia Chelini, Angela Di Capua, et al.Contrast Media & Molecular Imaging|October 11, 2019
Radiosynthesis and Preclinical Evaluation of 11C-VA426, a Cyclooxygenase-2 Selective LigandAssunta Carpinelli, Paolo Rainone, Sara Belloli, et al.Journal of Medicinal Chemistry|August 22, 2003
Synthesis, biological evaluation, and receptor docking simulations of 2-[(acylamino)ethyl]-1,4-benzodiazepines as kappa-opioid receptor agonists endowed with antinociceptive and antiamnesic activityMaurizio Anzini, Laura Canullo, Carlo Braile, et al.European Journal of Medicinal Chemistry|May 30, 2014
Synthesis and structure-activity relationship studies in serotonin 5-HT4 receptor ligands based on a benzo[de][2,6]naphthridine scaffoldFederica Castriconi, Marco Paolino, Germano Giuliani, et al.Bioorganic & Medicinal Chemistry|March 23, 2011
Non-peptide NK1 receptor ligands based on the 4-phenylpyridine moietyGermano Giuliani, Andrea Cappelli, Mario Matarrese, et al.Journal of Medicinal Chemistry|March 6, 2008
Design, synthesis, and biological evaluation of AT1 angiotensin II receptor antagonists based on the pyrazolo[3,4-b]pyridine and related heteroaromatic bicyclic systemsAndrea Cappelli, Chiara Nannicini, Andrea Gallelli, et al.Journal of Medicinal Chemistry|March 5, 2004
A non-peptide NK1 receptor agonist showing subpicomolar affinityAndrea Cappelli, Germano Giuliani, Gal la Pericot Mohr Gl, et al.Pageof 7