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Plos One|August 13, 2009
Activation of mGlu3 receptors stimulates the production of GDNF in striatal neuronsGiuseppe Battaglia, Gemma Molinaro, Barbara Riozzi, et al.Bioorganic & Medicinal Chemistry Letters|January 16, 2007
Chiral tetrahydroquinoline derivatives as potent anti-hyperalgesic agents in animal models of sustained inflammation and chronic neuropathic painRomano Di Fabio, Giuseppe Alvaro, Barbara Bertani, et al.Journal of Medicinal Chemistry|June 22, 2024
Discovery and Optimization of Pyridazinones as PI3Kδ Selective Inhibitors for Administration by InhalationPaolo Bruno, Alessandra Micoli, Mauro Corsi, et al.Neuropsychopharmacology : Official Publication of the American College of Neuropsychopharmacology|May 10, 2012
Role of orexin-1 receptor mechanisms on compulsive food consumption in a model of binge eating in female ratsLaura Piccoli, Maria Vittoria Micioni Di Bonaventura, Carlo Cifani, et al.Neuropharmacology|July 16, 2011
In vitro and in vivo characterization of the novel GABAB receptor positive allosteric modulator, 2-{1-[2-(4-chlorophenyl)-5-methylpyrazolo[1,5-a]pyrimidin-7-yl]-2-piperidinyl}ethanol (CMPPE)Elisabetta Perdona', Vivian J A Costantini, Michela Tessari, et al.Bioorganic & Medicinal Chemistry|October 1, 2013
Identification, biological characterization and pharmacophoric analysis of a new potent and selective NK1 receptor antagonist clinical candidateRomano Di Fabio, Giuseppe Alvaro, Simone Braggio, et al.Journal of Medicinal Chemistry|January 15, 2011
Discovery and biological characterization of (2R,4S)-1'-acetyl-N-{(1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethyl}-2-(4-fluoro-2-methylphenyl)-N-methyl-4,4'-bipiperidine-1-carboxamide as a new potent and selective neurokinin 1 (NK1) receptor antagonist clinical candidateRomano Di Fabio, Giuseppe Alvaro, Cristiana Griffante, et al.Journal of Medicinal Chemistry|April 25, 2009
Discovery process and pharmacological characterization of 2-(S)-(4-fluoro-2-methylphenyl)piperazine-1-carboxylic acid [1-(R)-(3,5-bis-trifluoromethylphenyl)ethyl]methylamide (vestipitant) as a potent, selective, and orally active NK1 receptor antagonistRomano Di Fabio, Cristiana Griffante, Giuseppe Alvaro, et al.Bioorganic & Medicinal Chemistry|June 22, 2011
Synthesis and structure-activity relationship of new 1,5-dialkyl-1,5-benzodiazepines as cholecystokinin-2 receptor antagonistsKaren Roberts, Antonella Ursini, Robert Barnaby, et al.Bioorganic & Medicinal Chemistry|December 10, 2002
Synthesis and pharmacological characterisation of 2,4-dicarboxy-pyrroles as selective non-competitive mGluR1 antagonistsFabrizio Micheli, Romano Di Fabio, Paolo Cavanni, et al.Pageof 6