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Bioorganic & Medicinal Chemistry Letters
|
April 20, 2005
Equipotent activity in both enantiomers of a series of ketopiperazine-based renin inhibitors
Noel A Powell, Emma H Clay, Daniel D Holsworth, et al.
Bioorganic & Medicinal Chemistry
|
December 8, 2004
The discovery and preparation of disubstituted novel amino-aryl-piperidine-based renin inhibitors
Wayne L Cody, Daniel D Holsworth, Noel A Powell, et al.
Bioorganic & Medicinal Chemistry
|
March 10, 2005
Discovery of novel non-peptidic ketopiperazine-based renin inhibitors
Daniel D Holsworth, Noel A Powell, Dennis M Downing, et al.
Bioorganic & Medicinal Chemistry Letters
|
April 30, 2013
Discovery of 2-((1H-benzo[d]imidazol-1-yl)methyl)-4H-pyrido[1,2-a]pyrimidin-4-ones as novel PKM2 activators
Chuangxing Guo, Angelica Linton, Mehran Jalaie, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 26, 2012
Design, synthesis, and evaluation of imidazo[4,5-c]pyridin-4-one derivatives with dual activity at angiotensin II type 1 receptor and peroxisome proliferator-activated receptor-γ
Agustin Casimiro-Garcia, Ronald J Heemstra, Christopher F Bigge, et al.
Bioorganic & Medicinal Chemistry Letters
|
May 8, 2007
Discovery of 6-ethyl-2,4-diaminopyrimidine-based small molecule renin inhibitors
Daniel D Holsworth, Mehran Jalaie, Thomas Belliotti, et al.
Analytical Biochemistry
|
November 23, 2006
Binding thermodynamics of substituted diaminopyrimidine renin inhibitors
Ronald W Sarver, Jeanette Peevers, Wayne L Cody, et al.
Journal of Medicinal Chemistry
|
May 12, 2011
Discovery of a series of imidazo[4,5-b]pyridines with dual activity at angiotensin II type 1 receptor and peroxisome proliferator-activated receptor-γ
Agustin Casimiro-Garcia, Gary F Filzen, Declan Flynn, et al.
Bioorganic & Medicinal Chemistry
|
June 19, 2007
Rational design of 6-(2,4-diaminopyrimidinyl)-1,4-benzoxazin-3-ones as small molecule renin inhibitors
Noel A Powell, Fred L Ciske, Cuiman Cai, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 17, 2006
Ketopiperazine-based renin inhibitors: optimization of the "C" ring
Daniel D Holsworth, Cuiman Cai, Xue-Min Cheng, et al.
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Showing results (11-20 of 27) with videos related to
Sort By:
Page
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Bioorganic & Medicinal Chemistry Letters
|
April 20, 2005
Equipotent activity in both enantiomers of a series of ketopiperazine-based renin inhibitors
Noel A Powell, Emma H Clay, Daniel D Holsworth, et al.
Bioorganic & Medicinal Chemistry
|
December 8, 2004
The discovery and preparation of disubstituted novel amino-aryl-piperidine-based renin inhibitors
Wayne L Cody, Daniel D Holsworth, Noel A Powell, et al.
Bioorganic & Medicinal Chemistry
|
March 10, 2005
Discovery of novel non-peptidic ketopiperazine-based renin inhibitors
Daniel D Holsworth, Noel A Powell, Dennis M Downing, et al.
Bioorganic & Medicinal Chemistry Letters
|
April 30, 2013
Discovery of 2-((1H-benzo[d]imidazol-1-yl)methyl)-4H-pyrido[1,2-a]pyrimidin-4-ones as novel PKM2 activators
Chuangxing Guo, Angelica Linton, Mehran Jalaie, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 26, 2012
Design, synthesis, and evaluation of imidazo[4,5-c]pyridin-4-one derivatives with dual activity at angiotensin II type 1 receptor and peroxisome proliferator-activated receptor-γ
Agustin Casimiro-Garcia, Ronald J Heemstra, Christopher F Bigge, et al.
Bioorganic & Medicinal Chemistry Letters
|
May 8, 2007
Discovery of 6-ethyl-2,4-diaminopyrimidine-based small molecule renin inhibitors
Daniel D Holsworth, Mehran Jalaie, Thomas Belliotti, et al.
Analytical Biochemistry
|
November 23, 2006
Binding thermodynamics of substituted diaminopyrimidine renin inhibitors
Ronald W Sarver, Jeanette Peevers, Wayne L Cody, et al.
Journal of Medicinal Chemistry
|
May 12, 2011
Discovery of a series of imidazo[4,5-b]pyridines with dual activity at angiotensin II type 1 receptor and peroxisome proliferator-activated receptor-γ
Agustin Casimiro-Garcia, Gary F Filzen, Declan Flynn, et al.
Bioorganic & Medicinal Chemistry
|
June 19, 2007
Rational design of 6-(2,4-diaminopyrimidinyl)-1,4-benzoxazin-3-ones as small molecule renin inhibitors
Noel A Powell, Fred L Ciske, Cuiman Cai, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 17, 2006
Ketopiperazine-based renin inhibitors: optimization of the "C" ring
Daniel D Holsworth, Cuiman Cai, Xue-Min Cheng, et al.
Page
of 3