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Bioorganic & Medicinal Chemistry Letters|March 5, 2018
Pyridazine and pyridazinone derivatives as potent and selective factor XIa inhibitorsZilun Hu, Cailan Wang, Wei Han, et al.Bioorganic & Medicinal Chemistry Letters|March 20, 2003
Nonbenzamidine isoxazoline derivatives as factor Xa inhibitorsMimi L Quan, Christopher D Ellis, Ming Y He, et al.Bioorganic & Medicinal Chemistry Letters|January 27, 2010
Phenyltriazolinones as potent factor Xa inhibitorsMimi L Quan, Donald J P Pinto, Karen A Rossi, et al.Bioorganic & Medicinal Chemistry Letters|February 5, 2003
Nonbenzamidine tetrazole derivatives as factor Xa inhibitorsMimi L Quan, Christopher D Ellis, Ming Y He, et al.Bioorganic & Medicinal Chemistry Letters|March 11, 2008
Sulfonamidolactam inhibitors of coagulation factor XaJoanne M Smallheer, Shuaige Wang, Mia L Laws, et al.Bioorganic & Medicinal Chemistry Letters|October 16, 2007
Design, structure-activity relationship, and pharmacokinetic profile of pyrazole-based indoline factor Xa inhibitorsJeffrey G Varnes, Dean A Wacker, Irina C Jacobson, et al.Bioorganic & Medicinal Chemistry Letters|January 17, 2015
Pyridine and pyridinone-based factor XIa inhibitorsJames R Corte, Tianan Fang, Jon J Hangeland, et al.Journal of Medicinal Chemistry|March 18, 2005
Discovery of 1-(3'-aminobenzisoxazol-5'-yl)-3-trifluoromethyl-N-[2-fluoro-4- [(2'-dimethylaminomethyl)imidazol-1-yl]phenyl]-1H-pyrazole-5-carboxyamide hydrochloride (razaxaban), a highly potent, selective, and orally bioavailable factor Xa inhibitorMimi L Quan, Patrick Y S Lam, Qi Han, et al.Journal of Medicinal Chemistry|January 14, 2017
Structure-Based Design of Macrocyclic Factor XIa Inhibitors: Discovery of the Macrocyclic Amide LinkerJames R Corte, Tianan Fang, Honey Osuna, et al.Bioorganic & Medicinal Chemistry Letters|September 12, 2006
Discovery of potent, efficacious, and orally bioavailable inhibitors of blood coagulation factor Xa with neutral P1 moietiesDonald J P Pinto, Robert A Galemmo, Mimi L Quan, et al.Pageof 3