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RSC Advances
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September 9, 2024
New <i>N</i>-phenylpyrrolamide inhibitors of DNA gyrase with improved antibacterial activity
Andrej Emanuel Cotman, Federica Fulgheri, Martina Piga, et al.
European Journal of Medicinal Chemistry
|
July 25, 2024
Development of narrow-spectrum topoisomerase-targeting antibacterials against mycobacteria
Maša Sterle, Eva Habjan, Martina Piga, et al.
Plos Biology
|
October 5, 2020
Rational design of balanced dual-targeting antibiotics with limited resistance
Akos Nyerges, Tihomir Tomašič, Martina Durcik, et al.
European Journal of Medicinal Chemistry
|
February 1, 2021
New dual ATP-competitive inhibitors of bacterial DNA gyrase and topoisomerase IV active against ESKAPE pathogens
Martina Durcik, Ákos Nyerges, Žiga Skok, et al.
European Journal of Medicinal Chemistry
|
September 5, 2024
Improved N-phenylpyrrolamide inhibitors of DNA gyrase as antibacterial agents for high-priority bacterial strains
Nace Zidar, Alessia Onali, Peter Peršolja, et al.
Bioorganic & Medicinal Chemistry
|
June 21, 2024
Exploring the interaction of N-(benzothiazol-2-yl)pyrrolamide DNA gyrase inhibitors with the GyrB ATP-binding site lipophilic floor: A medicinal chemistry and QTAIM study
Nace Zidar, Andrej Emanuel Cotman, Wessel Sinnige, et al.
Journal of Medicinal Chemistry
|
January 12, 2023
Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against <i>Acinetobacter baumannii</i> and <i>Pseudomonas aeruginosa</i>
Andrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, et al.
Journal of Medicinal Chemistry
|
March 6, 2023
New Dual Inhibitors of Bacterial Topoisomerases with Broad-Spectrum Antibacterial Activity and In Vivo Efficacy against Vancomycin-Intermediate <i>Staphylococcus aureus</i>
Martina Durcik, Andrej Emanuel Cotman, Žan Toplak, et al.
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of 8
Search research articles
Search
Showing results (71-80 of 78) with videos related to
Sort By:
Page
of 8
You have reached the last page of results.
This site can display upto 78 results.
RSC Advances
|
September 9, 2024
New <i>N</i>-phenylpyrrolamide inhibitors of DNA gyrase with improved antibacterial activity
Andrej Emanuel Cotman, Federica Fulgheri, Martina Piga, et al.
European Journal of Medicinal Chemistry
|
July 25, 2024
Development of narrow-spectrum topoisomerase-targeting antibacterials against mycobacteria
Maša Sterle, Eva Habjan, Martina Piga, et al.
Plos Biology
|
October 5, 2020
Rational design of balanced dual-targeting antibiotics with limited resistance
Akos Nyerges, Tihomir Tomašič, Martina Durcik, et al.
European Journal of Medicinal Chemistry
|
February 1, 2021
New dual ATP-competitive inhibitors of bacterial DNA gyrase and topoisomerase IV active against ESKAPE pathogens
Martina Durcik, Ákos Nyerges, Žiga Skok, et al.
European Journal of Medicinal Chemistry
|
September 5, 2024
Improved N-phenylpyrrolamide inhibitors of DNA gyrase as antibacterial agents for high-priority bacterial strains
Nace Zidar, Alessia Onali, Peter Peršolja, et al.
Bioorganic & Medicinal Chemistry
|
June 21, 2024
Exploring the interaction of N-(benzothiazol-2-yl)pyrrolamide DNA gyrase inhibitors with the GyrB ATP-binding site lipophilic floor: A medicinal chemistry and QTAIM study
Nace Zidar, Andrej Emanuel Cotman, Wessel Sinnige, et al.
Journal of Medicinal Chemistry
|
January 12, 2023
Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against <i>Acinetobacter baumannii</i> and <i>Pseudomonas aeruginosa</i>
Andrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, et al.
Journal of Medicinal Chemistry
|
March 6, 2023
New Dual Inhibitors of Bacterial Topoisomerases with Broad-Spectrum Antibacterial Activity and In Vivo Efficacy against Vancomycin-Intermediate <i>Staphylococcus aureus</i>
Martina Durcik, Andrej Emanuel Cotman, Žan Toplak, et al.
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