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Pharmaceuticals (Basel, Switzerland)|August 26, 2022
Improving Aqueous Solubility and In Vitro Pharmacokinetic Properties of the 3-Nitroimidazo[1,2-a]pyridine Antileishmanial PharmacophoreRomain Paoli-Lombardo, Nicolas Primas, Sandra Bourgeade-Delmas, et al.
Pharmaceuticals (Basel, Switzerland)|August 28, 2021
2-Phenoxy-3-Trichloromethylquinoxalines Are Antiplasmodial Derivatives with Activity against the Apicoplast of Plasmodium falciparumDyhia Amrane, Christophe-Sébastien Arnold, Sébastien Hutter, et al.
Chemical Biology & Drug Design|December 22, 2017
Design, synthesis, and antiprotozoal evaluation of new 2,9-bis[(substituted-aminomethyl)phenyl]-1,10-phenanthroline derivativesJean Guillon, Anita Cohen, Rabindra Nath Das, et al.
European Journal of Medicinal Chemistry|June 10, 2018
Novel 8-nitroquinolin-2(1H)-ones as NTR-bioactivated antikinetoplastid molecules: Synthesis, electrochemical and SAR studyJulien Pedron, Clotilde Boudot, Sébastien Hutter, et al.
European Journal of Medicinal Chemistry|March 21, 2015
Discovery of new thienopyrimidinone derivatives displaying antimalarial properties toward both erythrocytic and hepatic stages of PlasmodiumAnita Cohen, Peggy Suzanne, Jean-Charles Lancelot, et al.
European Journal of Medicinal Chemistry|August 10, 2018
8-Aryl-6-chloro-3-nitro-2-(phenylsulfonylmethyl)imidazo[1,2-a]pyridines as potent antitrypanosomatid molecules bioactivated by type 1 nitroreductasesCyril Fersing, Clotilde Boudot, Julien Pedron, et al.
ACS Medicinal Chemistry Letters|January 19, 2019
Nongenotoxic 3-Nitroimidazo[1,2-a]pyridines Are NTR1 Substrates That Display Potent in Vitro Antileishmanial ActivityCyril Fersing, Louise Basmaciyan, Clotilde Boudot, et al.
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