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Molecules (Basel, Switzerland)|January 20, 2021
A New CDK2 Inhibitor with 3-Hydrazonoindolin-2-One Scaffold Endowed with Anti-Breast Cancer Activity: Design, Synthesis, Biological Evaluation, and In Silico InsightsMohammad M Al-Sanea, Ahmad J Obaidullah, Mohamed E Shaker, et al.Bioorganic Chemistry|May 23, 2021
New bis([1,2,4]triazolo)[4,3-a:3',4'-c]quinoxaline derivatives as VEGFR-2 inhibitors and apoptosis inducers: Design, synthesis, in silico studies, and anticancer evaluationMohammed M Alanazi, Hazem A Mahdy, Nawaf A Alsaif, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|July 6, 2021
Design, synthesis, and analysis of antiproliferative and apoptosis-inducing activities of nitrile derivatives containing a benzofuran scaffold: EGFR inhibition assay and molecular modelling studySalma Fares, Khalid B Selim, Fatma E Goda, et al.Archiv Der Pharmazie|December 4, 2021
Targeting VEGFR-2 by new quinoxaline derivatives: Design, synthesis, antiproliferative assay, apoptosis induction, and in silico studiesNawaf A Alsaif, Hazem A Mahdy, Mohammed M Alanazi, et al.European Journal of Medicinal Chemistry|August 9, 2019
New anthranilic acid-incorporating N-benzenesulfonamidophthalimides as potent inhibitors of carbonic anhydrases I, II, IX, and XII: Synthesis, in vitro testing, and in silico assessmentAdel S El-Azab, Alaa A-M Abdel-Aziz, Silvia Bua, et al.Bioorganic Chemistry|March 18, 2019
Synthesis of benzensulfonamides linked to quinazoline scaffolds as novel carbonic anhydrase inhibitorsAdel S El-Azab, Alaa A-M Abdel-Aziz, Sivia Bua, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|February 4, 2020
Exploring structure-activity relationship of S-substituted 2-mercaptoquinazolin-4(3H)-one including 4-ethylbenzenesulfonamides as human carbonic anhydrase inhibitorsAdel S El-Azab, Alaa A-M Abdel-Aziz, Hany E A Ahmed, et al.Bioorganic Chemistry|September 8, 2019
Synthesis and comparative carbonic anhydrase inhibition of new Schiff's bases incorporating benzenesulfonamide, methanesulfonamide, and methylsulfonylbenzene scaffoldsAdel S El-Azab, Alaa A-M Abdel-Aziz, Silvia Bua, et al.Bioorganic Chemistry|March 29, 2019
Design, synthesis, and carbonic anhydrase inhibition activity of benzenesulfonamide-linked novel pyrazoline derivativesAlaa A-M Abdel-Aziz, Adel S El-Azab, Silvia Bua, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|March 20, 2020
S-substituted 2-mercaptoquinazolin-4(3H)-one and 4-ethylbenzensulfonamides act as potent and selective human carbonic anhydrase IX and XII inhibitorsAdel S El-Azab, Alaa A-M Abdel-Aziz, Silvia Bua, et al.Pageof 5